|
Alkylating analogs of peptide hormones. 1. Synthesis and properties of p-[N,N-bis(2-chloroethyl)amino]phenylbutyryl derivatives of bradykinin and bradykinin potentiating factor Richard J. Freer and John Morrow Stewart pp 1 - 5; DOI: 10.1021/jm00271a001 |
|
Alkylating analogs of peptide hormones. 2. Synthesis and properties of p-[N,N-bis(2-chloroethyl)amino]phenylbutyryl derivatives of angiotensin II Therezinha B. Paiva, Antonio C. M. Paiva, Richard J. Freer, and John Morrow Stewart pp 6 - 8; DOI: 10.1021/jm00271a002 |
|
Hypothalamic hormones. 27. Synthesis of di- and tripeptides and assay in vivo for activity in the thyrotropin releasing hormone and the luteinizing releasing hormone systems Hans Sievertsson, Jaw-Kang Chang, Karl Folkers, and Cyril Y. Bowers pp 8 - 11; DOI: 10.1021/jm00271a003 |
|
Solid phase synthesis of [3,4-dileucine]-oxytocin and a study of some of its pharmacological properties Myles A. Wille, Vincent Du Vigneaud, and W. Y. Chan pp 11 - 12; DOI: 10.1021/jm00271a004 |
|
Structural modification of S-trityl-L-cysteine. Preparation of some S-(substituted trityl)-L-cysteines and dipeptides of S-trityl-L-cysteine Kwang Yuen Zee-Cheng and C. C. Cheng pp 13 - 16; DOI: 10.1021/jm00271a005 |
|
Quantum mechanical study of the conformational properties of phenethylamines of biochemical and medicinal interest B. Pullman, J. L. Coubeils, Ph. Courriere, and J. P. Gervois pp 17 - 23; DOI: 10.1021/jm00271a006 |
|
Phenethylamine in a rigid framework. 2,3-Substituted cis- and trans-6-amino-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ols Bansi Lal, J. M. Khanna, and Nitya Anand pp 23 - 27; DOI: 10.1021/jm00271a007 |
|
Structure-activity relation studies on antimalarial phenanthrene amino alcohols. Modification of the side chain Ping-Lu Chien, Daniel J. McCaustland, William H. Burton, and C. C. Cheng pp 28 - 33; DOI: 10.1021/jm00271a008 |
|
Coenzyme Q. 139. Synthesis of new alkylamino- and alkylaminomethyl-5,8-quinolinequinones as inhibitors of coenzyme Q and as antimalarials Thomas H. Porter, Frederick S. Skelton, and Karl Folkers pp 34 - 36; DOI: 10.1021/jm00271a009 |
|
Mechanism of action of amodiaquine. Synthesis of its indoloquinoline analog Victor E. Marquez, Joseph W. Cranston, Raymond W. Ruddon, Lemont B. Kier, and Joseph H. Burckhalter pp 36 - 39; DOI: 10.1021/jm00271a010 |
|
Synthesis and biological activity of some 4-aryl-substituted 4-oxazolin-2-ones Francesco Bottari, Enrico Nannipieri, Marco F. Saettone, and Maria F. Serafini pp 39 - 42; DOI: 10.1021/jm00271a011 |
|
Derivatives of 4,5,-dihydro-1,3,-dimethyl-1H-pyrazolo[3,4-b][1,4]benzoxazepine with antiinflammatory activity Leo R. Swett, Robert G. Stein, and Eugene T. Kimura pp 42 - 45; DOI: 10.1021/jm00271a012 |
|
Cardiovascular drugs. 5. 1-Amino-3-phenoxy-2-propanol derivatives as .beta.-adrenergic blocking agents Michio Nakanishi, Tomio Muro, Yasuaki Chihara, Hiroshi Imamura, and Tooru Nakao pp 45 - 48; DOI: 10.1021/jm00271a013 |
|
.beta.-Adrenergic blocking agents. 11. Heterocycyclic analogs of pronethalol [2-isopropylamino-1-(2-naphthyl)ethanol] M. S. Chodnekar, A. F. Crowther, W. Hepworth, R. Howe, B. J. McLoughlin, A. Mitchell, B. S. Rao, R. P. Slatcher, L. H. Smith, and M. A. Stevens pp 49 - 57; DOI: 10.1021/jm00271a014 |
|
Potential renin inhibitors. 2. Ethanolamine and ethylamine derivatives of phospholipids Francis R. Pfeiffer, Clara K. Miao, Suzanne C. Hoke, and Jerry A. Weisbach pp 58 - 60; DOI: 10.1021/jm00271a015 |
|
Inhibitors of platelet aggregation. 3. {[(dialkylamino)alkyl]thio} heterocyclic compounds Edward F. Elslager, Neil F. Haley, J. R. McLean, Doris Potoczak, H. Veloso, and R. H. Wheelock pp 61 - 65; DOI: 10.1021/jm00271a016 |
|
Tumor inhibitors. 70. Structure-cytotoxicuty relations among N-acyltriamines related to solapalmitine S. Morris Kupchan, Goran Bondesson, and Alan P. Davies pp 65 - 68; DOI: 10.1021/jm00271a017 |
|
Mixed bifunctionality. 4. Antitumor activity of alkylating derivatives of polycyclic aromatic hydrocarbons as a function of structure and of vehicle Richard M. Peck and Anna P. O'Connell pp 68 - 70; DOI: 10.1021/jm00271a018 |
|
1,2-Disubstituted cyclopropane and cyclobutane derivatives related to acetylcholine Joseph G. Cannon, Arvind B. Rege, T. Lee Gruen, and John P. Long pp 71 - 75; DOI: 10.1021/jm00271a019 |
|
d1-.alpha.-(4-Cycloalkyl-1-cyclohexenyl)alkanoic acids and derivatives as antiinflammatory and antiarthritic compounds Michel Vincent, Georges Remond, and Jean C. Poignant pp 75 - 79; DOI: 10.1021/jm00271a020 |
|
Aminobenzoic acid diuretics. 3. 4-Substituted 5-sulfamylanthranilic acid derivatives Peter W. Feit and Ole B. Tvaermose Nielsen pp 79 - 83; DOI: 10.1021/jm00271a021 |
|
Preferred conformation of prostaglandin E1 James R. Hoyland and Lemont B. Kier pp 84 - 86; DOI: 10.1021/jm00271a022 |
|
C-3-Oxygenation of 17.alpha.-methyl-5.alpha.-androstan-17.beta.-o1 by rabbit liver homogenate Manfred E. Wolff and Yasuji Kasuya pp 87 - 88; DOI: 10.1021/jm00271a023 |
|
Synthesis and biological activity of D-bishomosteroids George Eadon and Carl Djerassi pp 89 - 91; DOI: 10.1021/jm00271a024 |
|
Cardiovascular activity of some substituted 2-aminobenzoquinolizines J. W. Van Dyke, H. J. Havera, R. D. Johnson, H. Vidrio, and A. Viveros pp 91 - 94; DOI: 10.1021/jm00271a025 |
|
N-carbalkoxy-O-alkylalkanamidoximes. New series of insecticides Dominick A. Coviello, Sheila L. Dvorin, and Bernard Greenberg pp 94 - 95; DOI: 10.1021/jm00271a026 |
|
Inhibition studies on antibody to poly(L-tyrosyl-L-glutamyl-L-alanylglycyl)glycine-1-14C ethyl ester. Synthesis and immunochemical properties of poly(L-alanyl-L-glutamy1-L-alanylglycyl)glycine-1-14C ethyl ester Brian J. Johnson, Charles Cheng, and Nora Tsang pp 95 - 97; DOI: 10.1021/jm00271a027 |
|
Synthesis of the trail marker of the Texas leaf-cutting ant, Atta texana Philip E. Sonnet pp 97 - 98; DOI: 10.1021/jm00271a028 |
|
Fibrin-stabilizing factor inhibitors. 4. Action of some synthetic fibrinoligase inhibitors on human platelet aggregation Ragnar Lunden, Ann Hartkoorn, J. Lars G. Nilsson, Pal Stenberg, Joyce Bruner-Lorand, and Laszlo Lorand pp 98 - 99; DOI: 10.1021/jm00271a029 |
|
Substituted thiazolidones and their selective inhibition of nicotinamide-adenine dinucleotide dependent oxidations Surendra S. Parmar, C. Dwivedi, A. Chaudhari, and T. K. Gupta pp 99 - 101; DOI: 10.1021/jm00271a030 |
|
Substituted thiazolylureas Peter J. Islip, Michael D. Closier, M. R. Johnson, and Martin C. Neville pp 101 - 103; DOI: 10.1021/jm00271a031 |
|
Antiviral benzimidazoles. Direct 1-substitution of 2-(.alpha.-hydroxybenzyl)benzimidazole and related compounds Desmond G. O'Sullivan and Anthony K. Wallis pp 103 - 104; DOI: 10.1021/jm00271a032 |
|
Secondary mechanisms of antifungal action of substituted 8-quinolinols. 3. 5,7,8-Substituted quinolines Herman Gerson, Maynard W. McNeil, Raulo Parmegiani, and Patricia K. Godfrey pp 105 - 106; DOI: 10.1021/jm00271a033 |
|
Heterocyclic compounds. 4. Synthesis and antiinflammatory activity of some substituted thienopyrimidones M. S. Manhas, S. D. Sharma, and S. G. Amin pp 106 - 107; DOI: 10.1021/jm00271a034 |
|
Antitumor activity of 2,2-hydrazobis(3-chloro-1,4-naphthoquinone) against Walker 256 (intramuscular) carcinosarcoma Benjamin Prescott pp 107 - 107; DOI: 10.1021/jm00271a035 |
|
Anthelmintic 2-(5-nitro-2-thienyl)-4-(substituted amino)quinazolines Robert J. Alaimo and Christopher J. Hatton pp 108 - 109; DOI: 10.1021/jm00271a036 |
|
Effects of S-(+)- and R-(-)-3,4,dimethoxyphenylisopropylamines in the rat Charles F. Barfknecht and David E. Nichols pp 109 - 110; DOI: 10.1021/jm00271a037 |
|
4-Amino-2-buten-1-o1 esters Robert E. Willette and Richard C. Driscoll pp 110 - 112; DOI: 10.1021/jm00271a038 |
|
Directional nature of hydrophobic bonding in phenethanolamine N-methyl transferase inhibitors Corwin Hansch and W. R. Glave pp 112 - 113; DOI: 10.1021/jm00271a039 |
|
N1,N1-Dialkyl-N4,N4-dialkylaminoacetylsulfanilamide as potent surface anesthetics I. Lalezari, A. Shafiee, M. A. Khoyi, and F. Abtahi pp 113 - 115; DOI: 10.1021/jm00271a040 |
|
Synthesis and antibacterial activity of 5-nitro-2-furfurylidene arylthioacethydrazides and 5-nitro-2-furfurylidene arylsulfonylacethydrazides I. Lalezari, P. Lowlavar, and N. Mazhari pp 115 - 116; DOI: 10.1021/jm00271a041 |
|
Acyl derivatives of 1-.beta.-D-arabinofuranosylcytosine John A. Montgomery and H. Jeanette Thomas pp 116 - 118; DOI: 10.1021/jm00271a042 |
|
Antibacterial activity of o-amino-N-hydroxybenzenesulfonamides Ned D. Heindel, C. C. Ho Ko, Richard B. Birrer, and Joseph R. Merkel pp 118 - 120; DOI: 10.1021/jm00271a043 |
|
5-Cyclohexyl-1-hydroxyacetylindans as potential antiinflammatory agents P. F. Juby, T. W. Hudyma, and R. A. Partyka pp 120 - 121; DOI: 10.1021/jm00271a044 |
|
Synthesis of some 6-hydroxymethyluracil derivatives K. L. Nagpal pp 121 - 122; DOI: 10.1021/jm00271a045 |
|
Synthesis of three oxytocin analogs related to [1-deaminopenicillamine]oxytocin prossessing antioxytocic activity Raymond J. Vavrek, Martha F. Ferger, G. Ashley Allen, Daniel H. Rich, Alfred T. Blomquist, and Vincent Du Vigneaud pp 123 - 126; DOI: 10.1021/jm00272a001 |
|
Role of the asparagine residue in oxytocin. Synthesis and biological properties of [5-.alpha.,.gamma.-diaminobutyric acid]oxytocin S. Hase, I. L. Schwartz, and R. Walter pp 126 - 128; DOI: 10.1021/jm00272a002 |
|
Synthesis and antiviral activities of adamantane spiro compounds. 1. Adamantane and analogous spiro-3'-pyrrolidines K. Lundahl, J. Schut, J. L. M. A. Schlatmann, G. B. Paerels, and A. Peters pp 129 - 132; DOI: 10.1021/jm00272a003 |
|
Synthesis and antiviral activities of adamantane spiro compounds. 2 R. Van Hes, A. Smit, T. Kralt, and A. Peters pp 132 - 136; DOI: 10.1021/jm00272a004 |
|
Biological inactivation of pyrrolnitrin. Identification and synthesis of pyrrolnitrin metabolites Patrick J. Murphy and Terry L. Williams pp 137 - 139; DOI: 10.1021/jm00272a005 |
|
Equilibrium and kinetic effects of sixteen compounds on the forms of horse heart ferricytochrome c George H. Czerlinski and Rita A. Galuszka pp 140 - 144; DOI: 10.1021/jm00272a006 |
|
Structure-activity correlations of antimalarial compounds. 1. Free-Wilson analysis of 2-phenylquinoline-4-carbinols Paul N. Craig pp 144 - 149; DOI: 10.1021/jm00272a007 |
|
Synthesis of 1-p-chlorobenzyl-7-azaindole-3-.alpha.-piperidylmethanol as a potential antimalarial agent Anthony J. Verbiscar pp 149 - 152; DOI: 10.1021/jm00272a008 |
|
Kinetics and mechanisms of drug action on microorganisms. 13. Comparative studies on action of lincomycin, clindamycin, and U 24729A against Escherichia coli Samuel M. Heman-Ackah and Edward R. Garrett pp 152 - 163; DOI: 10.1021/jm00272a009 |
|
Synthesis and biological activity of pyrazines and pyrazine ribonucleosides as pyrimidine analogs M. Bobek and A. Bloch pp 164 - 168; DOI: 10.1021/jm00272a010 |
|
Synthesis and biological activity of 4'-thio analogs of the antibiotic toyocamycin M. Bobek, R. L. Whistler, and A. Bloch pp 168 - 171; DOI: 10.1021/jm00272a011 |
|
Synthesis and antimicrobial activity of a carbocyclic puromycin analog. 6-Dimethylamino-9-[R-[2R-hydroxy-3R-(p-methoxyphenyl-L-alanylamino)]cyclopentyl]purine Susan Daluge and Robert Vince pp 171 - 177; DOI: 10.1021/jm00272a012 |
|
Identification and synthesis of the major nucleoside metabolite in rabbit urine after administration of puromycin aminonucleoside Herbert T. Nagasawa, Frances N. Shirota, and Carl S. Alexander pp 177 - 181; DOI: 10.1021/jm00272a013 |
|
Nucleosides of 2-azapurines and certain ring analogs John A. Montgomery and H. Jeanette Thomas pp 182 - 187; DOI: 10.1021/jm00272a014 |
|
N6-Substituted adenosines. Synthesis, biological activity, and some structure-activity relations M. H. Fleysher pp 187 - 191; DOI: 10.1021/jm00272a015 |
|
Potential antitumor agents. 5. Methylated .alpha.-(N)-heterocyclic carboxaldehyde thiosemicarbazones Krishna C. Agrawal, Robert J. Cushley, Seymour R. Lipsky, J. Randall Wheaton, and Alan C. Sartorelli pp 192 - 195; DOI: 10.1021/jm00272a016 |
|
Specificity of inhibition of coenzyme Q-enzyme systems by lipoidal benzoquinone derivatives Ronald S. Pardini, Joseph C. Catlin, James C. Heidker, and Karl Folkers pp 195 - 197; DOI: 10.1021/jm00272a017 |
|
.beta.-Adrenergic blocking agents of the chromone and xanthone groups P. Da Re, P. Valenti, A. Borraccini, and G. P. Primofiore pp 198 - 199; DOI: 10.1021/jm00272a018 |
|
Synthesis of trimethoprim variations. Replacement of methylene by polar groupings Eugene L. Stogryn pp 200 - 201; DOI: 10.1021/jm00272a019 |
|
Preparation and antitumor activity of derivatives of 1-phenyl-3,3-dimethyltriazene Ying-Tsung Lin, Ti Li Loo, Srikrishna Vadlamudi, and Abraham Goldin pp 201 - 203; DOI: 10.1021/jm00272a020 |
|
Synthesis of heterocyclic compounds. 438. Biochemical studies on drugs and the central nervous system. 1. Synthesis and activity of pyridoxal derivatives T. Kametani, M. Koizumi, K. Okui, Y. Nishii, and M. Ono pp 203 - 204; DOI: 10.1021/jm00272a021 |
|
Antimalarial compounds. 12. Guanidine derivatives of diphenyl sulfone and related compounds W. Peters, H. Piotrowska, B. Serafin, and T. Urbanski pp 204 - 206; DOI: 10.1021/jm00272a022 |
|
Synthesis and enzymological activity of 3-hydroxy-2-propyl-4,5-pyridinedimethanol Paul Melius and Joseph L. Greene pp 206 - 206; DOI: 10.1021/jm00272a023 |
|
Antimalarial activity and conformation of erythro- and threo-.alpha.-(2-piperidyl)-3,6-bis(trifluoromethyl)-9-phenanthrenemethanol R. E. Olsen pp 207 - 208; DOI: 10.1021/jm00272a024 |
|
N-Demethylation of morphine and structurally related compounds with chloroformate esters M. M. Abdel-Monem and P. S. Portoghese pp 208 - 210; DOI: 10.1021/jm00272a025 |
|
Synthesis of 4(3H)-pteridinones Ernst Felder, Davide Pitre, and Sergio Boveri pp 210 - 211; DOI: 10.1021/jm00272a026 |
|
Hepatocarcinogenicity of the trimethyl homologs of 4-dimethylaminoazobenzene Ellis V. Brown and Alice Kruegel pp 212 - 212; DOI: 10.1021/jm00272a027 |
|
Aliphatic amines as antipityrosporum agents Harold Dixon, Norman J. Van Abbe, and John K. Sugden pp 212 - 214; DOI: 10.1021/jm00272a028 |
|
Rapid, convenient preparative procedure for phenethylamines Edgar F. Kiefer pp 214 - 214; DOI: 10.1021/jm00272a029 |
|
Synthesis of 2-fluoro-9-.beta.-D-ribofuranosylpurine (2-fluoronebularine) Masajiro Kawana, Robert J. Rousseau, and Roland K. Robins pp 214 - 215; DOI: 10.1021/jm00272a030 |
|
4-[(Aminoxy)methyl]thiazole dihydrochloride Glenn H. Hamor pp 215 - 215; DOI: 10.1021/jm00272a031 |
|
Contractile Proteins and Muscle Alfred Burger pp 216 - 216; DOI: 10.1021/jm00272a900 |
|
Annual Reports in Medicinal Chemistry, 1970 Alfred Burger pp 216 - 216; DOI: 10.1021/jm00272a901 |
|
Narcotic Drugs. Biochemical Pharmacology Alfred Burger pp 216 - 216; DOI: 10.1021/jm00272a902 |
|
Lipid Metabolism Donald J. Hanahan pp 216 - 216; DOI: 10.1021/jm00272a903 |
|
Adrenocorticotropin. 40. Synthesis of a protected nonapeptide and of a biogically active nonadecapeptide related to adrenocorticotropic hormone. [5-Glutamine]adrenocorticotropin-(1-19) Choh Hao Li and Bahram Hemmasi pp 217 - 219; DOI: 10.1021/jm00273a001 |
|
Hypothalamic hormones. 32. Role of the histadine moiety in the structure of the thyrotropin-releasing hormone Hans Sievertsson, Jaw-Kang Chang, Karl Folkers, and Cyril Y. Bowers pp 219 - 221; DOI: 10.1021/jm00273a002 |
|
Hypothalamic hormones. 35. Two syntheses of the luteinizing hormone releasing hormone of the hypothalamus Hans Sievertsson, Jaw-Kang Chang, Alexander Von Klaudy, Conny Bogentoft, Bruce Currie, Karl Folkers, and Cyril Bowers pp 222 - 226; DOI: 10.1021/jm00273a003 |
|
Preliminary biological studies of several aliphatic amino acid analogs C. J. Abshire and G. Planet pp 226 - 229; DOI: 10.1021/jm00273a004 |
|
Irreversible enzyme inhibitors. 189. Inhibition of some dehydrogenases by derivatives of 4-hydroxyquinoline-2- and -3-carboxylic acids B. R. Baker and Ray R. Bramhall pp 230 - 233; DOI: 10.1021/jm00273a005 |
|
Irreversible enzyme inhibitors. 190. Inhibition of some dehydrogenases by 1-substituted-1,4-dihydro-4-quinolone-3-carboxylic acids B. R. Baker and Ray R. Bramhall pp 233 - 235; DOI: 10.1021/jm00273a006 |
|
Irreversible enzyme inhibitors. 191. Hydrophobic bonding to some dehydrogenases by 6-, 7-, or 8-substituted-4-hydroxyquinoline-3-carboxylic acids B. R. Baker and Ray R. Bramhall pp 235 - 237; DOI: 10.1021/jm00273a007 |
|
Irreversible enzyme inhibitors. 192. Hydrophobic bonding to some dehydrogenases with 5-substituted-4-hydroxyquinoline-3-carboxylic acids B. R. Baker and Ray R. Bramhall pp 237 - 241; DOI: 10.1021/jm00273a008 |
|
Conformational aspects of systems related to acetylcholine. 3. Base-catalyzed and acetycholinesterase-catalyzed hydrolysis of the isomeric dl-3-trimethylammonium-2-acetoxy-trans-decalin halides and the isomeric dl-1-methyl-3-acetoxy-trans-decahydroquinoline methiodides William F. Stephen, Edward E. Smissman, Katherine B. Schowen, and Gary W. Self pp 241 - 243; DOI: 10.1021/jm00273a009 |
|
Structural parameters determining cholinergic and anticholinergic activities in a series of 1,3-dioxolanes K. J. Chang, R. C. Deth, and D. J. Triggle pp 243 - 247; DOI: 10.1021/jm00273a010 |
|
Medicinal chemical studies on antiplasmin drugs. 4. Chemical modification of trans-4-aminomethylcyclohexanecarboxylic acid and its effect on antiplasmin activity Atsuji Okano, Masato Inaoko, Shoichi Funabashi, Masahiro Iwamoto, Sumiro Isoda, Reimei Moroi, Yasushi Abiko, and Miyoshi Hirata pp 247 - 255; DOI: 10.1021/jm00273a011 |
|
Potential antileukemic and immunosuppressive drugs. 3. Effects of homocyclic ring substitution on the in vitro drug activity of 4-nitrobenzo-2,1,3-oxadiazoles (4-nitrobenzofurazans) and their N-oxides (4-nitrobenzofuroxans) P. B. Ghosh, B. Ternai, and M. W. Whitehouse pp 255 - 260; DOI: 10.1021/jm00273a012 |
|
.beta.-Adrenergic blocking agents. 12. Heterocyclic compounds related to propranolol A. F. Crowther, R. Howe, B. J. McLoughlin, K. B. Mallion, B. S. Rao, L. H. Smith, and R. W. Turner pp 260 - 266; DOI: 10.1021/jm00273a013 |
|
Synthesis and biological activity of acronycine analogs J. Schneider, E. L. Evans, E. Grunberg, and Ian R. Fryer pp 266 - 270; DOI: 10.1021/jm00273a014 |
|
Metabolism of 1-[(5-nitrofurfurylidene)amino]-2-imidazolidinone Donald L. Pugh, Joanne Olivard, Harry R. Snyder, and James P. Heotis pp 270 - 273; DOI: 10.1021/jm00273a015 |
|
Centrally acting emetics. 5. Preparation and pharmacology of 10-hydroxy-11-methoxyaporphine (Isoapocodeine). In vitro enzymic methylation of apomorphine Joseph G. Cannon, Robert V. Smith, Ali Modiri, S. Paul Sood, Robert J. Borgman, Mohd. A. Aleem, and John Paul Long pp 273 - 276; DOI: 10.1021/jm00273a016 |
|
Antiviral agents. 5H-as-Triazino[5,6-b]indoles Jan M. Z. Gladych, Roy Hornby, John H. Hunt, David Jack, John J. Boyle, Robert J. Ferlauto, Richard F. Haff, Charles G. Kormendy, Fredrick J. Stanfield, and Richard C. Stewart pp 277 - 281; DOI: 10.1021/jm00273a017 |
|
Anthelmintic activity in sheep of some compounds related to pyrantel and morantel W. C. Austin, R. L. Cornwell, R. M. Jones, and M. Robinson pp 281 - 285; DOI: 10.1021/jm00273a018 |
|
Agents acting on the central nervous system. 14. 1-(p-alkanoylphenoxy)-3-(N4-arylpiperazinyl)propan-2-ols. New class of antidepressants S. Nivas Rastogi, Nitya Anand, and C. R. Prasad pp 286 - 291; DOI: 10.1021/jm00273a019 |
|
Local anesthetic activity of 2-piperazinecarboxanilides Walter L. McKenzie and William O. Foye pp 291 - 295; DOI: 10.1021/jm00273a020 |
|
Bicyclic Mannich bases. 1. Psychotropic activity of 2-(4-aryl-l-piperazinyl)bicyclo[3.3.1]nonan-9-ones and derivatives Robert N. Schut, Frederick E. Ward, and Rodolfo Rodriguez pp 301 - 304; DOI: 10.1021/jm00273a021 |
|
Nucleosides of 8-azapurines .nu.-triazolo[4,5-d]pyrimidines) John A. Montgomery and H. Jeanette Thomas pp 305 - 307; DOI: 10.1021/jm00273a022 |
|
Glutathione. 6. Probable mechanism of action of diazene antibiotics Edward M. Kosower and Tetsuo Miyadera pp 307 - 312; DOI: 10.1021/jm00273a023 |
|
Organic disulfides and related substances. 33. Sodium 4-(2-acetamidoethyldithio)butanesulfinate and related compounds as antiradiation drugs Lamar Field and Yong H. Khim pp 312 - 315; DOI: 10.1021/jm00273a024 |
|
Insect chemosterilants. 11. Substituted 3,5-diamino-1,2,4-dithiazolium salts and related compounds J. E. Oliver, S. C. Chang, R. T. Brown, J. B. Stokes, and A. B. Borkovec pp 315 - 320; DOI: 10.1021/jm00273a025 |
|
Molecular weight studies on the active constituents of compound 48/80 George W. Read and James F. Lenney pp 320 - 323; DOI: 10.1021/jm00273a026 |
|
Synthesis of 5-hydroxymethyl-, 5-acetoxymethyl-, and 5-methylmercapto-7,12-dimethylbenz[a]anthracenes, and of 5,7,12-trimethylbenz[a]anthracene Melvin S. Newman and Robert F. Cunico pp 323 - 325; DOI: 10.1021/jm00273a027 |
|
Preparation and antimicrobial properties of the D and L forms of 3-amino-3,4-dihydro-1-hydroxycarbostyril Alvie L. Davis, David R. Smith, David C. Foyt, Janet L. Black, and Tommy J. McCord pp 325 - 327; DOI: 10.1021/jm00273a028 |
|
Inhibition of dopamine .beta.-hydroxylase by 5-phenoxymethyl-2-oxazolidinethiones G. A. Johnson, E. G. Kim, S. J. Boukma, D. Lednicer, and G. A. Youngdale pp 327 - 329; DOI: 10.1021/jm00273a029 |
|
Preparation of a camoquin derivative with quaternary carbon side chain P. N. Natarajan and Ngiam Tong Lan pp 329 - 330; DOI: 10.1021/jm00273a030 |
|
Hill reaction inhibitors. 3. Conformational aspects of ureas Sharon G. Boots, Marvin R. Boots, and Donald E. Moreland pp 330 - 332; DOI: 10.1021/jm00273a031 |
|
Bicyclic triazoles. 1. 3-(2-Furyl)-5-phenylthiazolo-[2,3-c]-s-triazole Man M. Kochhar and B. B. Williams pp 332 - 333; DOI: 10.1021/jm00273a032 |
|
Antibacterial activity of 6-(5-membered heteroarylacetamido)penicillanic acids Ronald G. Micetich, Rintje Raap, John Howard, and Imre Pushkas pp 333 - 335; DOI: 10.1021/jm00273a033 |
|
Antibacterial 2,3-dihydro-2-(5-nitro-2-thienyl)quinazolin-4-(1H)-ones Robert J. Alaimo and H. Eric Russell pp 335 - 336; DOI: 10.1021/jm00273a034 |
|
DL-1-(.alpha.-Methylbenzyl)-2-methylimidazole-5-carboxylate esters. Synthesis and pharmacological properties Erik F. Godefroi and J. Th. J. Platje pp 336 - 337; DOI: 10.1021/jm00273a035 |
|
Cysteine scavengers. 1. Bis(3-pyridylmethyl) phosphate and bis(3-pyridylmethyl) pyrophosphate Mervyn Israel, Marilyn A. Whitesell, Edward J. Modest, George E. Foley, Herbert Lazarus, and Franz Bergel pp 337 - 338; DOI: 10.1021/jm00273a036 |
|
Cobalt derivatives of Schiff bases of aliphatic amines as antitumor agents Ernest M. Hodnett and William J. Dunn pp 339 - 339; DOI: 10.1021/jm00273a037 |
|
Improved synthesis of the antibiotic, hexahydrospinamycin Tetsuo Miyadera and Edward M. Kosower pp 339 - 340; DOI: 10.1021/jm00273a038 |
|
Triphenylpropylpiperazine Derivatives as New Potent Analgetic Substances G.L. Regnier, R. J. Canevari, J. C. Le Douarec, S. Holstorp, and J. Daussy pp 295 - 301; DOI: 10.1021/jm00273a600 |
|
Inhibition of adrenal phenethanolamine-N-methyltransferase by substituted imidazoles N. P. Jensen, S. M. Schmitt, T. B. Windholz, T. Y. Shen, L. R. Mandel, B. Lopez-Ramos, and C. C. Porter pp 341 - 344; DOI: 10.1021/jm00274a001 |
|
Lowering of serum lipid levels by "masked" nicotinic acid derivatives Denis M. Bailey, David Wood, Robert E. Johnson, John P. McAuliff, James C. Bradford, and Aaron Arnold pp 344 - 348; DOI: 10.1021/jm00274a002 |
|
Centrally acting emetics. 6. Derivatives of .beta.-naphthylamine and 2-indanamine Joseph G. Cannon, Jack C. Kim, Mohd. A. Aleem, and John Paul Long pp 348 - 350; DOI: 10.1021/jm00274a003 |
|
Schistosomicides. 2. Derivatives of 2,3,4,4a,5,6-hexahydro-1H-pyrazino[1,2-.alpha.]quinoline C. A. R. Baxter and H. C. Richards pp 351 - 356; DOI: 10.1021/jm00274a004 |
|
Structure of hydroxycotinine, a nicotine methobolite Ermias Dagne and Neal Castagnoli pp 356 - 360; DOI: 10.1021/jm00274a005 |
|
(+)-6,6-Difluoronorgestrel, A New synthetic hormonal steroid Alexander L. Johnson pp 360 - 363; DOI: 10.1021/jm00274a006 |
|
Steroid side-chain oxazolidines Eugene J. Agnello and Peter R. Farina pp 363 - 365; DOI: 10.1021/jm00274a007 |
|
Novel anthelmintic agents. 6. Pyrantel analogs with activity against whipworm James W. McFarland and Horold L. Howes pp 365 - 368; DOI: 10.1021/jm00274a008 |
|
Heterocyclic steroids. 4. Synthesis and androgenic activity of A-ring homosteroids Galal Zanati and Manfred E. Wolff pp 368 - 369; DOI: 10.1021/jm00274a009 |
|
Naphthothiophenes. 1. .alpha.-(Alkylaminomethyl)-4-naphtho[2,1-b]thiophenemethanols as antimalarials B. P. Das, J. A. Campbell, F. B. Samples, R. A. Wallace, L. K. Whisenant, R. W. Woodard, and D. W. Boykin pp 370 - 374; DOI: 10.1021/jm00274a010 |
|
Influence of stereochemistry and lipophilicity on biological activity of some ganglionic blocking agents Robert A. Wiley, Bahjat A. Faraj, Allen Jantz, and Milos M. Hava pp 374 - 378; DOI: 10.1021/jm00274a011 |
|
Antistaphylococcal and antifibrinolytic activities of N.alpha.-(.omega.-aminoacyl)-L-lysines Akira Fujii, Kinji Tanaka, and Elton S. Cook pp 378 - 380; DOI: 10.1021/jm00274a012 |
|
Analogs of S-adenosylhomocysteine as potential inhibitors of biological transmethylation. Synthesis and biological activity of homocysteine derivatives bridged to adenine James K. Coward and William D. Sweet pp 381 - 384; DOI: 10.1021/jm00274a013 |
|
Conformation of gastrin tetrapeptide Lemont B. Kier and Jack M. George pp 384 - 386; DOI: 10.1021/jm00274a014 |
|
Platelet aggregation inhibitors. 2. Inhibition of platelet aggregation by 5'-, 2-, 6-, and 8-substituted adenosines Kiyomi Kikugawa, Kazuhiro Iizuka, Yoshiyuki Higuchi, Hachihiko Hirayama, and Motonobu Ichino pp 387 - 390; DOI: 10.1021/jm00274a015 |
|
Rates of alkaline hydrolysis and muscarinic activity of some aminoacetates and their quaternary ammonium analogs A. K. Cho, D. J. Jenden, and S. I. Lamb pp 391 - 394; DOI: 10.1021/jm00274a016 |
|
Correlation of antihypertensive activity with structure in a series of 2H-1,2,4-benzothiadiazine 1,1-dioxides using the substituent constant approach John G. Topliss and Milton D. Yudis pp 394 - 400; DOI: 10.1021/jm00274a017 |
|
.pi.-Substituent constants for the 2H-1,2,4-benzothiadiazine 1,1-dioxide system John G. Topliss and Milton D. Yudis pp 400 - 403; DOI: 10.1021/jm00274a018 |
|
Conformations of highly hindered aryl ethers. 10. Intramolecular aryl-iodine .pi. complex formation and its relation to thyromimetic activity Pedro A. Lehmann pp 404 - 409; DOI: 10.1021/jm00274a019 |
|
Synthesis and oral hypoglycemic activity of N-(p-deuteriomethylbenzenesulfonyl)-N'-n-butylurea, deuterium-substituted tolbutamide Raymond D. Kimbrough pp 409 - 410; DOI: 10.1021/jm00274a020 |
|
Polymers containing phenethylamines Ben-Zion Weiner, Menashe Tahan, and Albert Zilkha pp 410 - 413; DOI: 10.1021/jm00274a021 |
|
Potential psychotomimetics. New bromoalkoxyamphetamines Silvia Sepulveda, Ricardo Valenzuela, and Bruce K. Cassels pp 413 - 415; DOI: 10.1021/jm00274a022 |
|
1H-Imidazo[1,2-.alpha.]imidazoles Laird F. Miller and Ronald E. Bambury pp 415 - 417; DOI: 10.1021/jm00274a023 |
|
Synthesis and central nervous system activity of new piperazine derivatives. 4 J. A. Fernandez, R. A. Bellare, C. V. Deliwala, N. K. Dadkar, and U. K. Sheth pp 417 - 419; DOI: 10.1021/jm00274a024 |
|
Heterocycles. 5. Oxazole N-oxides P. M. Weintraub pp 419 - 420; DOI: 10.1021/jm00274a025 |
|
Antiviral agents. 2. Analogs of 2-(.alpha.-hydroxybenzyl)benzimidazole F. Gualtieri, G. Brody, A. H. Fieldsteel, and W. A. Skinner pp 420 - 422; DOI: 10.1021/jm00274a026 |
|
Conformation dependency of antibody to poly(L-tyrosyl-L-glutamyl-L-alanylglycyl)glycine-l-14C ethyl ester Brian J. Johnson pp 423 - 424; DOI: 10.1021/jm00274a027 |
|
exo-Bicyclo[3.1.0]hexane-6-carboxylic acid and related compounds, oral hypoglycemic agents Ronald H. Rynbrandt, Fred E. Dutton, and Fredericka L. Schmidt pp 424 - 426; DOI: 10.1021/jm00274a028 |
|
Estradiol analogs with conformational flexibility. 4-(1,2,3,4-Tetrahydro-6-'ydroxy-2-naphthyl)butan-2-ol P. Narasimha Rao, David H. Buss, and Leonard R. Axelrod pp 426 - 427; DOI: 10.1021/jm00274a029 |
|
Ornithine analogs as potential ornithine decarboxylase inhibitors. 1. N-Substituted ornithine derivatives W. A. Skinner and J. G. Johansson pp 427 - 428; DOI: 10.1021/jm00274a030 |
|
Molecular orbital calculations on the preferred conformation of neostigmine James W. Crow and William C. Holland pp 429 - 429; DOI: 10.1021/jm00274a031 |
|
Acylpyruvates as potential antifungal agents Homer Burch and Joseph E. Gray pp 429 - 431; DOI: 10.1021/jm00274a032 |
|
Biologically oriented organic sulfur chemistry. 10. Inhibitory effects of certain organic sulflur compounds on Histoplasma capsulatum Ilda McVeigh, Susan Evans, Lamar Field, Wayne S. Hanley, and C. Emory Tate pp 431 - 433; DOI: 10.1021/jm00274a033 |
|
Quinoxaline studies. 20. Potential antimalarials. Synthesis of anti- and syn-N,N-dialkylaminomethyl 2-quinoxalinyl ketoximes Henry R. Moreno, John E. Oatis, and Harry P. Schultz pp 433 - 434; DOI: 10.1021/jm00274a034 |
|
Potential antidiabetics. 11. Preparation of 4-arylazo-3,5-disubstituted-(2H)-1,2,6-thiadiazine 1,1-dioxides H. G. Garg and Chandra Prakash pp 435 - 436; DOI: 10.1021/jm00274a035 |
|
Potential antitumor agent dicyclohexylammonium 2-[4-[N,N-bis(2-chloroethyl)amino]phenoxy]-2-methylpropionate Harold Z. Sommer and George E. Wicks pp 436 - 437; DOI: 10.1021/jm00274a036 |
|
Structure-activity studies on sulfamyl diuretics Perter W. Feit, Ole B. T. Nielsen, and Herta Bruun pp 437 - 440; DOI: 10.1021/jm00274a037 |
|
4-Anilino-1-phenyl-3-pyrrolecarboxylic acids. Analogs of the fenamic acids Victor J. Bauer and S. R. Safir pp 440 - 441; DOI: 10.1021/jm00274a038 |
|
Derivatives of 9-amino-9H-purine-6(1H)-thione Carroll Temple, Conrad L. Kussner, and John A. Montgomery pp 441 - 442; DOI: 10.1021/jm00274a039 |
|
Pyrido[2,3-d]pyrimidine-6-carboxamides as potential diuretic agents Arthur A. Santilli and Dong Han Kim pp 442 - 443; DOI: 10.1021/jm00274a040 |
|
Synthesis and antiarrhythmic activity of some N-(adamantylaminoalkyl)benzamides V. L. Narayanan and F. J. Sweeney pp 443 - 445; DOI: 10.1021/jm00274a041 |
|
Cyclic derivatives of 2-cyclohexylamino-1-phenylethanol W. J. Irwin, D. L. Wheeler, and N. J. Harper pp 445 - 446; DOI: 10.1021/jm00274a042 |
|
Central nervous system, antidiuretic, and some other activities of pyrazoles H. G. Garg pp 446 - 447; DOI: 10.1021/jm00274a043 |
|
3,3'-Ethylenediglutarimide as a potential tumor inhibitor David B. Haydock and Thomas P. C. Mulholland pp 447 - 448; DOI: 10.1021/jm00274a044 |
|
Preparation of tumor-specific boron compounds. 1. In vitro studies using boron-labeled antibodies and elemental boron as neutron targets M. Frederick Hawthorne, Richard J. Wiersema, and Mitsuo Takasugi pp 449 - 452; DOI: 10.1021/jm00275a001 |
|
Quantum-mechanical study of the conformational properties of sympatholytic compounds J. L. Coubeils, Ph. Courriere, and B. Pullman pp 453 - 455; DOI: 10.1021/jm00275a002 |
|
Enzyme inhibitors. 25. Equation to calculate the unknown Ki from two known values of Ki in an R,S, and RS series. Stereoselectivity of inhibition of adenosine deaminase by (R)-, (S)-, and (RS)-9-(1-hydroxy-2-alkyl and -aralkyl)adenines Howard J. Schaeffer, R. N. Johnson, Michael A. Schwartz, and Charles F. Schwender pp 456 - 458; DOI: 10.1021/jm00275a003 |
|
Accumulation of cyclic adenosine monophosphate in incubated slices of brain tissue. 1. Structure-activity relation of agonists and antagonists of biogenic amines and of tricyclic tranquilizers and antidepressants Minta Huang and John W. Daly pp 458 - 462; DOI: 10.1021/jm00275a004 |
|
Accumulation of cyclic adenosine monophosphate in incubated slices of brain tissue. 2. Effects of depolarizing agents, membrane stabilizers, phosphodiesterase inhibitors, and adenosine analogs Minta Huang, Hirotoshi Shimizu, and John W. Daly pp 462 - 466; DOI: 10.1021/jm00275a005 |
|
Relation between antihistamine and antidepressant activity in hexahydroindenopyridines J. Augstein, A. L. Ham, and P. R. Leeming pp 466 - 470; DOI: 10.1021/jm00275a006 |
|
Heterocyclic O-substituted hydroxylamines. Antiinflammatory activity and possible inhibition of histamine biosynthesis Glenn H. Hamor and Fulvio Rubessa pp 470 - 471; DOI: 10.1021/jm00275a007 |
|
Pyrimidine derivatives and related compounds. 15. Synthesis and analgetic and antiinflammatory activities of 1,3-substituted 5-amino-6-methyluracil derivatives Shigeo Senda, Kosaku Hirota, and Kazuo Banno pp 471 - 476; DOI: 10.1021/jm00275a008 |
|
Psychosedative agents. 2. 8-(4-Substituted 1-piperazinylalkyl)-8-azaspiro[4.5]decane-7,9-diones Yao-Hua Wu, J. W. Rayburn, L. E. Allen, H. C. Ferguson, and J. W. Kissel pp 477 - 479; DOI: 10.1021/jm00275a009 |
|
Synthetic thyrotropin-releasing factor analogs. 3. Effect of replacement or modification of histidine residue on biological activity J. Rivier, W. Vale, M. Monahan, N. Ling, and R. Burgus pp 479 - 482; DOI: 10.1021/jm00275a010 |
|
Synthesis of 1-hydroxy-L-proline and related cyclic N-hydroxyamino acids. Metabolic disposition of carbon-14-labeled 1-hydroxy-L-proline in rodents H. T. Nagasawa, J. G. Kohlhoff, P. S. Fraser, and A. A. Mikhail pp 483 - 486; DOI: 10.1021/jm00275a011 |
|
Synthesis and certain pharmacological properties of lysine-vasopressinoic acid methylamide and lysine-vasopressinoic acid dimethylamide John D. Glass and Vincent Du Vigneaud pp 486 - 488; DOI: 10.1021/jm00275a012 |
|
Immunochemical studies on linear antigenic polypeptides with a known primary structure. Specificity of antibodies to poly(L-tyrosyl-L-glutamyl-L-alanylglycyl)glycine-1-14C ethyl ester Brian J. Johnson and Nora Tsang pp 488 - 490; DOI: 10.1021/jm00275a013 |
|
Antimalarials. 1. 2-Quinolinemethanols A. Markovac, C. L. Stevens, and A. B. Ash pp 490 - 493; DOI: 10.1021/jm00275a014 |
|
Stereochemical studies on medicinal agents. 11. Metabolism and distribution of prodine isomers in mice M. M. Abdel-Monem, D. L. Larson, H. J. Kupferberg, and P. S. Portoghese pp 494 - 500; DOI: 10.1021/jm00275a015 |
|
Synthesis of .alpha.-[p-(fluoren-9-ylidenemethyl) phenyl]-2-piperidineethanol, an inhibitor of platelet aggregation George P. Claxton, J. Martin Grisar, Edward M. Roberts, and Robert W. Fleming pp 500 - 504; DOI: 10.1021/jm00275a016 |
|
Coenzyme Q. 147. Synthesis of new 2-alkylamino-1,4-naphthoquinones as inhibitors of coenzyme Q and as antimalarials Thomas H. Porter, Frederick S. Skelton, Christine M. Bowman, and Karl Folkers pp 504 - 506; DOI: 10.1021/jm00275a017 |
|
Stereochemical studies of antimuscarinic agents. Diastereoisomeric esters of 3-tropanol, 1,3-dimethyl-4-piperidinol, and related compounds D. F. Biggs, A. F. Casy, and W. K. Jeffery pp 506 - 509; DOI: 10.1021/jm00275a018 |
|
Compounds affecting the central nervous system. 2. Aromatic acetals of tropanediols Sol. J. Daum, Anthony J. Gambino, Mario D. Aceto, and Robert L. Clarke pp 509 - 514; DOI: 10.1021/jm00275a019 |
|
Diazirines. 3. Synthesis of a series of diazirine-containing molecules and their pharmacological evaluation Robert F. R. Church, Raymond R. Maleike, and Martin J. Weiss pp 514 - 518; DOI: 10.1021/jm00275a020 |
|
4-Oxo-1,2,3,4-tetrahydroquinazolines. 3. Synthesis and choleretic activity of quinazoline derivatives Kentaro Okumura, Yoshihisa Yamada, Toyonari Oine, Junichi Tani, Takashi Ochiai, and Ichizo Inoue pp 518 - 523; DOI: 10.1021/jm00275a021 |
|
Basic ethers of 2-anilinobenzothiazoles and 2-anilinobenzoxazoles as potential antidepressants C. J. Sharpe, P. J. Palmer, D. E. Evans, G. R. Brown, Gillian King, R. S. Shadbolt, R. B. Trigg, R. J. Ward, A. Ashford, and Janet W. Ross pp 523 - 529; DOI: 10.1021/jm00275a022 |
|
Diuretics. 1. 1-Imidoyl-2-(2- and 3-indolyl)indolines Yao-Hua Wu, Walter G. Lobeck, Richard P. Ryan, and Allen W. Gomoll pp 529 - 534; DOI: 10.1021/jm00275a023 |
|
Receptor site labeling through functional groups. 2. Reactivity of maleimide groups Tetsuo Miyadera and Edward M. Kosower pp 534 - 537; DOI: 10.1021/jm00275a024 |
|
Sulfamoyl azides. Hydrolysis rates and hypotensive activity W. L. Matier, W. T. Comer, and D. Deitchman pp 538 - 541; DOI: 10.1021/jm00275a025 |
|
Biotransformation of the antiarrhythmic agent 1-[o[[3-(dimethylamino)propyl]thio]phenyl]-3-methylurea in the dog Allen I. Cohen, Jacques Dreyfuss, and Henry M. Fales pp 542 - 545; DOI: 10.1021/jm00275a026 |
|
Conformational aspects of systems related to acetylcholine. 4. Syntheses of the dl-2-dimethylamino-trans-decalin methiodides Edward E. Smissman, Ronald T. Borchardt, and Katharine B. Schowen pp 545 - 548; DOI: 10.1021/jm00275a027 |
|
Spirans. 19. Spirans with functional groups Leonard M. Rice, Bhagvandas S. Sheth, and Theodore B. Zalucky pp 548 - 551; DOI: 10.1021/jm00275a028 |
|
Antiinflammatory 2,3-dihydro-2-oxobenzofuran-3-carboxanilides Saul B. Kadin pp 551 - 552; DOI: 10.1021/jm00275a029 |
|
Substituted anilides of 3-monoethyl ester of 4-hydroxyisophthalic acid R. Spano, G. Linari, and R. Marri pp 552 - 553; DOI: 10.1021/jm00275a030 |
|
Substituted thiazolidones as anticonvulsants C. Dwivedi, T. K. Gupta, and Surendra S. Parmar pp 553 - 554; DOI: 10.1021/jm00275a031 |
|
Synthesis of N'-substituted arylsulfonylpyrazoles, their anthelmintic activity, and the cytotoxicity of some hydrazides H. G. Garg and Narendrajit Kaur pp 554 - 555; DOI: 10.1021/jm00275a032 |
|
Preparation and progestational activity of 6-cyano-16-methylene-17.alpha.-hydroxy-4,6-pregnadiene-3,20-dione 17-acetate and related compounds T. L. Popper, H. P. Faro, F. E. Carlon, and H. L. Herzog pp 555 - 556; DOI: 10.1021/jm00275a033 |
|
Antiinflammatory activities of 17,21-methyl ortho esters, 17-mono- and 17,21-diesters of 6.alpha.,9.alpha.-difluorocorticosteroids R. Gardi, R. Vitali, G. Falconi, and A. Ercoli pp 556 - 558; DOI: 10.1021/jm00275a034 |
|
Pyrido[3,2-g]pteridines. 1. Chemistry and growth-inhibitory activity of some 1H,3H-2,4-dioxopyrido[3,2-g]pteridines (9-azaaloxazines Mervyn Israel, Lynne C. Jones, and Edward J. Modest pp 558 - 561; DOI: 10.1021/jm00275a035 |
|
Nucleoside peptides. 4. Synthesis of certain 1-(N-4-aminoacyl-4-amino-2,3-4-trideoxy-.beta.-D-erythro-hex-2-enopyranuronic acid) cytosine derivatives related to blasticidin S Masajiro Kawana, David G. Streeter, Robert J. Rousseau, and Roland K. Robins pp 561 - 564; DOI: 10.1021/jm00275a036 |
|
Mixed thiolsulfonates and sulfonamides from polyfunctional mercaptans using trifluoromethyl thiosulfonates James P. Weidner and Seymour S. Block pp 564 - 567; DOI: 10.1021/jm00275a037 |
|
Synthesis and biologic evaluation of 7-hydroxymethotrexate, 7-methylaminopterin, and 7-methylmethotrexate David Farquhar, Ti Li Loo, and Srikrishna Vadlamudi pp 567 - 569; DOI: 10.1021/jm00275a038 |
|
Synthesis of 5-fluoro-6,8-dimethylbenz[a] anthracene Melvin S. Newman, Joseph H. Cecil, and William M. Hung pp 569 - 570; DOI: 10.1021/jm00275a039 |
|
2-Pyrazinecarboxanilides Walter L. McKenzie and William O. Foye pp 570 - 571; DOI: 10.1021/jm00275a040 |
|
2,5-Anhydro-1-deoxy-1-[(6-methylthio)purin-9-yl]-D-allitol John A. Montgomery and Kathleen Hewson pp 571 - 571; DOI: 10.1021/jm00275a041 |
|
Book Reviews pp 572 - 572; DOI: 10.1021/jm00275a600 |
|
Interrelation of the regression models used for structure-activity analyses Arthur Cammarata pp 573 - 577; DOI: 10.1021/jm00276a001 |
|
Structure-activity relations among some antiinflammatory 3-(5-aryl-2-tetrazolyl)alkanoic acids and derivatives Robert T. Buckler pp 578 - 583; DOI: 10.1021/jm00276a002 |
|
Synthesis and structure-activity relations of disodium cromoglycate and some related compounds H. Cairns, C. Fitzmaurice, D. Hunter, P. B. Johnson, J. King, T. B. Lee, G. H. Lord, R. Minshull, and J. S. G. Cox pp 583 - 589; DOI: 10.1021/jm00276a003 |
|
Synthesis and analgetic activity of 1,2-disubstituted 2-phenylethylamines Arturo Donetti, Ernesta Marazzi-Uberti, Silvano Cadadio, and Camillo Bianchi pp 590 - 592; DOI: 10.1021/jm00276a004 |
|
Bridged compounds as potential analgetics. Substituted 3-exo-dimethylaminomethylnorbornanes as potential analgetics. Syntheses and stereochemistry of some 2-hydroxy-2-aryl substituted 3-exo-dimethylaminomethylnorbornanes A. H. Beckett, V. Nacci, and Abdul Q. Khokhar pp 593 - 594; DOI: 10.1021/jm00276a005 |
|
N-Alicyclic-substituted derivatives of 2-aminoethanethiol and related compounds as antiradiation agents Robert D. Elliott, James R. Piper, Carl R. Stringfellow, and Thomas P. Johnston pp 595 - 600; DOI: 10.1021/jm00276a006 |
|
Optically active dithiothreitol. Toxicity and radiation-protective activity Marvin Carmack, Charles J. Kelley, Steadman D. Harrison, and Kenneth P. DuBois pp 600 - 603; DOI: 10.1021/jm00276a007 |
|
General anesthetics. 3. Fluorinated methyl ethyl ethers as anesthetic agents Ross C. Terrell, Louise Speers, Alex J. Szur, Thomas Ucciardi, and James F. Vitcha pp 604 - 606; DOI: 10.1021/jm00276a008 |
|
General anesthetics. 4. Methyl pentahaloethyl and methyl heptahaloisopropyl ethers as anesthetic agents Louise Speers, Alex J. Szur, and Ross C. Terrell pp 606 - 608; DOI: 10.1021/jm00276a009 |
|
Antitumor agents. 3. Synthesis and cytotoxic activity of helenalin amine adducts and related derivatives Kuo-Hsiung Lee, Hiroshi Furukawa, and Eng-Shang Huang pp 609 - 611; DOI: 10.1021/jm00276a010 |
|
Potential antitumor agents. 12. 9-Anilinoacridines G. J. Atwell, B. F. Cain, and R. N. Seelye pp 611 - 615; DOI: 10.1021/jm00276a011 |
|
Potential antitumor agents. 8. Derivatives of 3- and 5-benzyloxy-2-formylpyridine thiosemicarbazone Ai Jeng Lin, Krishna C. Agrawal, and Alan C. Sartorelli pp 615 - 618; DOI: 10.1021/jm00276a012 |
|
Tumor inhibitors. 3. Identification and synthesis of a oncolytic hydrocarbon from American coneflower roots Denys J. Voaden and Martin Jacobson pp 619 - 623; DOI: 10.1021/jm00276a013 |
|
Hypothalamic hormones. 36. Synthesis of the luteinizing-releasing hormone of the hypothalamus and the 8-lysine analog Jaw-Kang Chang, Hans Sievertsson, Bruce L. Currie, Conny Bogentoft, Karl Folkers, and Cyril Y. Bowers pp 623 - 627; DOI: 10.1021/jm00276a014 |
|
Solid-phase synthesis of [6-arginine]-,[4-histidine, 6-tyrosine]-, and [8-isoleucine]angiotensins II Mahesh C. Khosla, Satyendra Jumar, Robert R. Smeby, and F. Merlin Bumpus pp 627 - 629; DOI: 10.1021/jm00276a015 |
|
Synthesis and properties of 1-deamino-8-L-homolysine-vasopressin Gunnar Lindeberg, Jaroslav Kyncl, Patricia Dreyfuss, and Miklos Bodanszky pp 629 - 631; DOI: 10.1021/jm00276a016 |
|
Chemical modifications of erythromycin antibiotics. 3. Synthesis of 4'' and 11 esters of erythromycin A and B Peter H. Jones, Thomas J. Perun, Elizabeth K. Rowley, and Evelyn J. Baker pp 631 - 634; DOI: 10.1021/jm00276a017 |
|
Chemical modification of erythromycin antibiotics. 4. Structure-activity relations of erythromycin esters Yvonne C. Martin, Peter H. Jones, Thomas J. Perun, Walton E. Grudy, Stanley Bell, Robert R. Bower, and Nathan L. Shipkowitz pp 635 - 638; DOI: 10.1021/jm00276a018 |
|
Irreversible enzyme inhibitors. 193. Inhibition of choline acetyltransferase,, Mode of binding by 4-stilbazoles B. R. Baker and Raymond E. Gibson pp 639 - 642; DOI: 10.1021/jm00276a019 |
|
Synthesis and pharmacological evaluation of some .beta.,.beta.-disubstituted analogs of acetylcholine D. F. Biggs, A. F. Casy, I. Chu, and R. T. Coutts pp 642 - 646; DOI: 10.1021/jm00276a020 |
|
Acetylcholinesterase reactivators. Pyridyl and anilyl trifluoromethyl ketoximes R. L. Salvador, M. Saucier, D. Simon, and R. Goyer pp 646 - 650; DOI: 10.1021/jm00276a021 |
|
.beta.-Adrenergic blocking agents. 3-(3-Substituted-amino-2-hydroxypropoxy)-4-substituted-1,2,5-thiadiazoles B. K. Wasson, W. K. Gibson, R. S. Stuart, H. W. R. Williams, and C. H. Yates pp 651 - 655; DOI: 10.1021/jm00276a022 |
|
Bisbenzimidazoles. Potent inhibitors of rhinoviruses William R. Roderick, Carl W. Nordeen, Anne M. Von Esch, and Raynor N. Appell pp 655 - 658; DOI: 10.1021/jm00276a023 |
|
Hypocholesterolemic indole-2-carboxylic acids Takashi Kariya, J. Martin Grisar, Norbert L. Wiech, and Thomas R. Blohm pp 659 - 662; DOI: 10.1021/jm00276a024 |
|
Synthesis and biological activity of some 5-substituted 2,4-diamino-6-alkylpyrimidines. 3 James P. Jonak, Sigmund F. Zakrzewski, and Lawrence H. Mead pp 662 - 665; DOI: 10.1021/jm00276a025 |
|
Analogs of phenothiazines. 4. Effect of structure upon neuropharmacological activity of some chlorpromazine analogs of the diphenylmethane type Carl Kaiser, Alex M. Pavloff, Eleanor Garvey, Philip J. Fowler, David H. Tedeschi, Charles L. Zirkle, Edward A. Nodiff, and Andrew J. Saggiomo pp 665 - 673; DOI: 10.1021/jm00276a026 |
|
Fibrin-stabilizing factor inhibitors. 5. Primary amines related to monotosylcadaverine Pal Stenberg, Christine Ljunggren, J. L. G. Nilsson, Ragnar Lunden, and Olle Eriksson pp 674 - 675; DOI: 10.1021/jm00276a027 |
|
Fluorinated pyrimidines. 41. Syntheses of 5-trifluoromethyl-3'-deoxyuridine and 5-fluoro-3'-deoxyuridine Stephen Nesnow, A. Mohsin Mian, Toshikazu Oki, Daniel L. Dexter, and Charles Heidelberger pp 676 - 677; DOI: 10.1021/jm00276a028 |
|
3,5-Disubstituted-6-methyl-2-pyridone. Dihydrazide, dicarbamate, and monoaminoalkyl ester Brian Jaques and John W. Hubbard pp 677 - 678; DOI: 10.1021/jm00276a029 |
|
Preparation and progestational activity of 6-trifluoromethyl-16-methylene-17.alpha.-hydroxy-4,6-pregnadiene-3,20-dione 17-acetate and related compounds H. P. Faro, R. E. Youngstrom, T. L. Popper, R. Neri, and H. L. Herzog pp 679 - 681; DOI: 10.1021/jm00276a030 |
|
Specificity in enzyme inhibition. 2. .alpha.-Aminohydroxamic acids as inhibitors of histidine decarboxylase and 3,4-dihydroxyphenylalanine decarboxylase Edward E. Smissman and Victor D. Warner pp 681 - 682; DOI: 10.1021/jm00276a031 |
|
Adamantyl analogs of the antidepressive, 5-(2-dimethylaminoethyl)-2,3-dihydro-2-phenyl-1,5-benzothiazepin-4(5H))-one V. L. Narayanan pp 682 - 684; DOI: 10.1021/jm00276a032 |
|
4,6-Didemethyl-4,6-dibromoactinomycin C1 (D) Frank Seela pp 684 - 686; DOI: 10.1021/jm00276a033 |
|
Syntheses of heterocyclic compounds. 459. Synthesis of rescinnamine-like compounds as antihypertensive agents T. Kametani, M. Ihara, T. Suzuki, T. Takahashi, R. Iwaki, H. Takei, N. Miyake, M. Yoshida, Y. Hasegawa, and H. Kitagawa pp 686 - 687; DOI: 10.1021/jm00276a034 |
|
Analgetics based on the pyrrolidine ring. 7 Ian M. Lockhart, Nigel E. Webb, Michael Wright, Claude W. Winder, and Mary A. Hare pp 687 - 690; DOI: 10.1021/jm00276a035 |
|
Synthesis of new glycido derivatives. 2-Dimethylaminoethyl triphenylglycidate and 2-dimethylaminoethyl 2,3,3-triphenylglycidyl ether Arturo Donetti and Bruno Lumachi pp 690 - 690; DOI: 10.1021/jm00276a036 |
|
Alkyl derivatives of tetrahydroisoquinoline, 1-phenylpiperazine, and 4-diphenylmethylpiperidine W. J. Irwin, D. L. Wheeler, and N. J. Harper pp 690 - 692; DOI: 10.1021/jm00276a037 |
|
1-(4-Dimethylaminoethoxy-3-methoxyphenyl)-2-aminoalkanes Marta A. Colombini and Alfred Burger pp 692 - 693; DOI: 10.1021/jm00276a038 |
|
1,4-Disubstituted piperazines. 3. Piperazinylbenzothiazoles Matthew Verderame pp 693 - 694; DOI: 10.1021/jm00276a039 |
|
Synthesis of 1,2,4-triazoles as potential hypoglycemic agents Benjamin Blank, Diana M. Nichols, and Praful D. Vaidya pp 694 - 696; DOI: 10.1021/jm00276a040 |
|
Solid-phase synthesis of seryltyrosylserylmethionylglutaminylhistidylphenylalanylarginyltryptophylglycine hydrazide and its N.alpha.-tert-butyloxycarbonyl derivative and their melanotropic activity Choh Hao Li and Bahram Hemmasi pp 697 - 699; DOI: 10.1021/jm00277a001 |
|
Sulfonamide structure-activity relation in a cell-free system. Correlation of inhibition of folate synthesis with antibacterial activity and physicochemical parameters G. H. Miller, P. H. Doukas, and J. K. Seydel pp 700 - 706; DOI: 10.1021/jm00277a002 |
|
Pharmacokinetics, metabolism, and urinary excretion of [3H]-alphaprodine in dogs M. M. Abdel-Monem, P. A. Harris, and P. S. Portoghese pp 706 - 708; DOI: 10.1021/jm00277a003 |
|
Metabolites of probenecid. Chemical, physical, and pharmacological studies Z. H. Israili, J. M. Perel, R. F. Cunningham, P. G. Dayton, T. F. Yu, A. B. Gutman, K. R. Long, R. C. Long, and J. H. Goldstein pp 709 - 713; DOI: 10.1021/jm00277a004 |
|
.alpha.,.alpha.'-and B,.beta.'-Deuterium-labeled dopamine. Synthesis and pharmacologic actions J. M. Perel, D. K. Dawson, P. G. Dayton, and L. I. Goldberg pp 714 - 716; DOI: 10.1021/jm00277a005 |
|
Synthesis and biological activity of 17-esters of 6-dehydro-16-methylene-17.alpha.-hydroxyprogesterones E. L. Shapiro, L. Weber, H. Harris, C. Miskowicz, R. Neri, and H. L. Herzog pp 716 - 720; DOI: 10.1021/jm00277a006 |
|
1-Phenyl-2-phenethyl-1,2,3,4-tetrahydroisoquinolines. New series of nonsteroidal female antifertility agents Rolf Paul, John A. Coppola, and Elliott Cohen pp 720 - 726; DOI: 10.1021/jm00277a007 |
|
Amidines. 2. New class of antihypertensive agents. 1,2,3,5-Tetrahydroimidazo[2,1-b]quinazolines Timothy Jen, Barbara Dienel, Helene Bowman, John Petta, Anna Helt, and Bernard Loev pp 727 - 731; DOI: 10.1021/jm00277a008 |
|
Synthetic antibacterials. 4. Nitrofurylvinylpyrido[2,3-d]pyrimidine derivatives Sadao Nishigaki, Kazuko Ogiwara, Shinobu Fukazawa, Misuzu Ichiba, Noriko Mizushima, and Fumio Yoneda pp 731 - 734; DOI: 10.1021/jm00277a009 |
|
Synthesis and biological activity of selected 2,6-disubstituted(2-deoxy-.alpha.- and -.beta.-D-erythro-pentofuranosyl)purines Leon F. Christensen, Arthur D. Broom, Morris J. Robins, and Alexander Bloch pp 735 - 739; DOI: 10.1021/jm00277a010 |
|
Antitumor and mutagenic properties of a variety of heterocyclic nitrogen and sulfur mustards Hugh J. Creech, Robert K. Preston, Richard M. Peck, Anna P. O'Connell, and Bruce N. Ames pp 739 - 746; DOI: 10.1021/jm00277a011 |
|
Medicinal chemistry of [10] annulenes and related compounds. 1. 11-Azatricyclo[4.4.1.01,6]undecane, 11-azatricyclo[4.4.1.01,6]undeca-3,8-diene, and 11-azabicyclo[4.4.1]undeca-1,3,5,7,9-pentaene as antiviral agents Gary L. Grunewald, Ann M. Warner, Sheryl J. Hays, Robert H. Bussell, and Marilyn K. Seals pp 747 - 750; DOI: 10.1021/jm00277a012 |
|
Derivatives of 10,11-dihydro-5H-dibenzo[a,d]cycloheptene and related compounds. 6. Aminoalkyl derivatives of the aza isosteres Frank J. Villani, Peter J. L. Daniels, Claire A. Ellis, Thomas A. Mann, Kai-Chih Wang, and Elizabeth A. Wefer pp 750 - 754; DOI: 10.1021/jm00277a013 |
|
Synthesis of fatty acids with smooth muscle stimulant activity. 3. Acetylenic analogs of 12-hydroxyheptadeca-trans-8,trans-10-dienoic acid E. Crundwell and A. L. Cripps pp 754 - 756; DOI: 10.1021/jm00277a014 |
|
Fluorescent derivatives of strophanthidin. Interaction with sodium- and potassium-activated adenosine triphosphatase Franz Oesch, James A. Waters, John W. Daly, and Bernhard Witkop pp 757 - 759; DOI: 10.1021/jm00277a015 |
|
Sulfur and selenium compounds related to acetylcholine and choline. 11. Selenocarbonyl ester and selenocarboxamide analogs of local anesthetics Shih-Hsi Chu, Gilbert R. Hillman, and Henry G. Mautner pp 760 - 762; DOI: 10.1021/jm00277a016 |
|
N-Phenyl-2-indolinones and N-phenylindolines. New class of antidepressant agents A. Canas-Rodriguez and P. R. Leeming pp 762 - 770; DOI: 10.1021/jm00277a017 |
|
Antimalarial arylaminopropanols W. T. Colwell, V. Brown, P. Christie, J. Lange, C. Reece, K. Yamamoto, and D. W. Henry pp 771 - 775; DOI: 10.1021/jm00277a018 |
|
Antimalarial phenanthrene amino alcohols. 2. Trifluoromethyl-containing 9-phenanthrenemethanols Edward A. Nodiff, Andrew J. Saggiomo, Masafu Shinbo, Eugene H. Chen, Hirotaka Otomasu, Yasuaki Kondo, Toyohiko Kikuchi, Basant L. Verma, Shin Matsuura, and et al. pp 775 - 780; DOI: 10.1021/jm00277a019 |
|
Experimentally induced phenylketonuria. 4. Potential inhibitors of phenylalanine hydroxylase Joseph I. DeGraw, Vernon H. Brown, W. A. Skinner, Susan LeValley, and Chozo Mitoma pp 781 - 781; DOI: 10.1021/jm00277a020 |
|
Steroids and related natural products. 70. Conversion of cardenolides to isocardanolides F. Warren Villaescusa and George R. Pettit pp 781 - 783; DOI: 10.1021/jm00277a021 |
|
Synthesis and antiinflammatory activity of betamethasone 17-benzoate A. Ercoli, G. Falconi, R. Gardi, and R. Vitali pp 783 - 784; DOI: 10.1021/jm00277a022 |
|
6,6-Difluoro-19-norprogesterone Alexander L. Johnson pp 784 - 785; DOI: 10.1021/jm00277a023 |
|
Book Reviews pp 785 - 786; DOI: 10.1021/jm00277a600 |
|
Binding of apolar molecules by serum albumin J. M. Vandenbelt, Corwin Hansch, and C. Church pp 787 - 789; DOI: 10.1021/jm00278a001 |
|
Nucleic acids. 13. 3'-0- and 2'-0-esters of 1-.beta.-D-arabinofuranosylcytosine as antileukemic and immunosuppressive agents Donald T. Warner, Gary L. Neil, Arlen J. Taylor, and William J. Wechter pp 790 - 792; DOI: 10.1021/jm00278a002 |
|
Synthesis of some analogs of angiotensin II as specific antagonists of the parent hormone M. C. Khosla, R. A. Leese, W. L. Maloy, A. T. Ferreira, R. R. Smeby, and F. M. Bumpus pp 792 - 795; DOI: 10.1021/jm00278a003 |
|
Sulfur analogs of dopamine and norepinephrine. Inhibition of catechol-O-methyltransferase W. B. Lutz, C. R. Creveling, J. W. Daly, B. Witkop, and L. I. Goldberg pp 795 - 802; DOI: 10.1021/jm00278a004 |
|
Cis- and trans-2-mercaptocyclobutylamines. Synthesis and antilipolytic properties in vitro Donald T. Witiak, Birandra K. Sinha, Ock Soon Lee, and Dennis R. Feller pp 803 - 808; DOI: 10.1021/jm00278a005 |
|
Antimalarials. 2. 2,6-Bis(aryl)-4-pyridinemethanols P. Blumbergs, M. P. LaMontagne, A. Markovac, J. G. Moehring, A. B. Ash, and C. L. Stevens pp 808 - 812; DOI: 10.1021/jm00278a006 |
|
Antimalarial drugs. 24. Folate antagonists. 2. 2,4-Diamino-6-{[aralkyl and (heterocyclic)methyl]amino}quinazolines, a novel class of antimetabolites of interest in drug-resistant malaria and Chagas' disease John Davoll, A. M. Johnson, H. J. Davies, O. D. Bird, J. Clarke, and Edward F. Elslager pp 812 - 826; DOI: 10.1021/jm00278a007 |
|
Antimalarial drugs. 25. Folate antagonists. 3. 2,4-Diamino-6-(heterocyclic)quinazolines, a novel class of antimetabolites with potent antimalarial and antibacterial activity Edward F. Elslager, J. Clarke, Leslie M. Werbel, Donald F. Worth, and John Davoll pp 827 - 836; DOI: 10.1021/jm00278a008 |
|
Antimalarial substances. 26. Folate antagonists. 4. Antimalarial and antimetabolite effects of 2,4-diamino-6-[(benzyl)amino]pyrido[2,3-d]pyrimidines John Davoll, J. Clarke, and Edward F. Elslager pp 837 - 839; DOI: 10.1021/jm00278a009 |
|
5'-O-methyl derivatives of 1-.beta.-D-arabinofuranosylcytosine and 1-.beta.-D-arabinofuranosyluracil Jerzy Giziewicz, Jaroslaw T. Kusmierek, and David Shugar pp 839 - 840; DOI: 10.1021/jm00278a010 |
|
Cotinine N-oxide, a new metabolite of nicotine Ermias Dagne and Neal Castagnoli pp 840 - 841; DOI: 10.1021/jm00278a011 |
|
Azapurine nucleosides. 3. Synthesis of 7-(.beta.-D-ribofuranosyl)imidazo[4,5-d]-.gamma.-triazin-4-one (2-azainosine) and related derivatives Masajiro Kawana, George A. Ivanovics, Robert J. Rousseau, and Roland K. Robins pp 841 - 843; DOI: 10.1021/jm00278a012 |
|
Transformations in the morphine series. 5. Reaction of codeinone with dimethyloxosulfonium methylide. Structure and analgetic activity of the product and its reduced form Lewis J. Sargent and Arthur E. Jacobson pp 843 - 845; DOI: 10.1021/jm00278a013 |
|
Alkaloids in mammalian tissues. 2. Synthesis of (+)- and (-)-1-substituted-6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolines S. Teitel, J. O'Brien, and A. Brossi pp 845 - 846; DOI: 10.1021/jm00278a014 |
|
Anticonvulsant activity of nitrobenzamides and their inhibition of nicotinamide-adenine dinucleotide dependent oxidations Surendra S. Parmar, C. Dwivedi, Basheer Ali, and R. S. Misra pp 846 - 848; DOI: 10.1021/jm00278a015 |
|
Sudoxicam and related N-heterocyclic carboxamides of 4-hydroxy-2H-1,2-benzothiazine 1,1-dioxide. Potent nonsteroidal antiinflammatory agents Joseph G. Lombardino and Edward H. Wiseman pp 848 - 849; DOI: 10.1021/jm00278a016 |
|
Antineoplastic activity of 6-dimethylaminonicotinamide Leland R. Lewis and C. C. Cheng pp 849 - 850; DOI: 10.1021/jm00278a017 |
|
2-Phenyl-4H-cyclopentathiazole-4-carboxylic acids as potential antiinflammatory agents Francis J. McEvoy and George R. Allen pp 850 - 851; DOI: 10.1021/jm00278a018 |
|
Synthesis and central nervous system depressant activity of new oxaza heterocyclic amides G. Pifferi, P. Consonni, A. Diena, and B. Rosselli Del Turco pp 851 - 853; DOI: 10.1021/jm00278a019 |
|
Chemistry of adamantane. 5. Synthesis and anticholinergic properties of 1-adamant-1-yl-1-phenyl-3-N-pyrrolidino-1-propanol hydrochloride Colin H. Cashin, Terrence M. Hotten, and Stephen S. Szinai pp 853 - 854; DOI: 10.1021/jm00278a020 |
|
17.alpha.-Propadienyl, 17.alpha.-propynyl, and 17.alpha.-trifluoropropynyl analogs of 6,6-difluoronorethindrone Alexander L. Johnson pp 854 - 855; DOI: 10.1021/jm00278a021 |
|
Convenient synthesis of 1,1-disubstituted 1,4-butanediols and derivatives Suminori Umio, Ikuo Ueda, and Hiroshi Nojima pp 855 - 856; DOI: 10.1021/jm00278a022 |
|
Synthesis and anthelmintic activity of some sulfonylbenzimidazoles R. D. Haugwitz, B. V. Maurer, and V. L. Narayanan pp 856 - 858; DOI: 10.1021/jm00278a023 |
|
Antimalarial activities of some 3,5-diamino-as-triazine derivatives Richard W. A. Rees, Peter B. Russell, Theodore J. Foell, and Royal E. Bright pp 859 - 861; DOI: 10.1021/jm00278a024 |
|
Synthesis of halogenated anthraldehydes and their conversion to antimalarial amino alcohols James T. Traxler, E. Patrick Lira, and Clarence W. Huffman pp 861 - 863; DOI: 10.1021/jm00278a025 |
|
3-Chromanamine hydrochlorides with central stimulant activity Ian M. Lockhart and Sheila A. Foard pp 863 - 865; DOI: 10.1021/jm00278a026 |
|
Benzopyrones. 7. Synthesis and antiallergic activity of some 2-(5-tetrazolyl)chromones G. P. Ellis and D. Shaw pp 865 - 867; DOI: 10.1021/jm00278a027 |
|
Photochemistry of zearalenone and its derivatives C. Allan Peters pp 867 - 868; DOI: 10.1021/jm00278a028 |
|
.beta.-Adrenergic blocking agents of the chromone and xanthone groups. II. Propanolol type derivatives P. Da Re, G. P. Primofiore, and A. Bertelli pp 868 - 869; DOI: 10.1021/jm00278a029 |
|
Preparation of N-(2-chloroethyl)-N-(2-hydroxyethyl)arylamines. Possible intermediates to potential carcinolytic agents bearing dissimilar reactive functions Allan B. Foster, Michael Jarman, Walter C. J. Ross, and Michael J. Tisdale pp 869 - 870; DOI: 10.1021/jm00278a030 |
|
.omega.-(N,N-diethylamino)-n-alkyl 3,4,5-trimethoxybenzoates as local anesthetics Casey P. Robinson and B. V. Rama Sastry pp 870 - 872; DOI: 10.1021/jm00278a031 |
|
Antitumor activity of some derivatives of daunorubicin at the amino and methyl ketone functions Kazuko Yamamoto, Edward M. Acton, and David W. Henry pp 872 - 875; DOI: 10.1021/jm00278a032 |
|
Mannich bases of 2,3-dihydro-4(1H)-carbazolones as potential psychotropic agents Ruddy Littell, E. N. Greenblatt, and George R. Allen pp 875 - 876; DOI: 10.1021/jm00278a033 |
|
Synthesis of some spin-labeled analogs of drug molecules Colin F. Chignell, Donnas K. Starkweather, and Ronald H. Erlich pp 876 - 878; DOI: 10.1021/jm00278a034 |
|
Azapurine nucleosides. 1. Synthesis and antitumor activity of certain 3-.beta.-D-ribofuranosyl- and 2'-deoxy-D-ribofuranosyl-v-triazolo[4,5-d]pyrimidines Wolfgang Hutzenlaub, Richard L. Tolman, and Roland K. Robins pp 879 - 883; DOI: 10.1021/jm00279a001 |
|
Azapurine nucleosides. 2. Synthesis and antiviral activity of 7-amino-3-.alpha.-D-arabinofuranosyl-v-triazolo[4,5-d]pyrimidine and related nucleosides Clive W. Smith, Robert W. Sidwell, Roland K. Robins, and Richard L. Tolman pp 883 - 887; DOI: 10.1021/jm00279a002 |
|
2,5-Dihydro-1,2,4-benzothiadiazepine 1,1-dioxides. Synthesis and pharmacological evaluation M. P. Fernandez-Tome, R. Madronero, J. Del Rio, and S. Vega pp 887 - 890; DOI: 10.1021/jm00279a003 |
|
Synthesis and pharmacological properties of 3-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-ylidene)-1,2-dialkylpyrrolidine derivatives Suminori Umio, Masahiro Hitomi, Hiroshi Nojima, Noriyuki Kumadaki, Ikuo Ueda, Tadamasa Kanaya, and Yoshio Deguchi pp 891 - 894; DOI: 10.1021/jm00279a004 |
|
[3H]-Vincristine. Preparation and preliminary pharmacology Richard J. Owellen and Douglas W. Donigian pp 894 - 898; DOI: 10.1021/jm00279a005 |
|
Stability of some phenothiazine free radicals Louis Levy, Thomas N. Tozer, L. Dallas Tuck, and Donald B. Loveland pp 898 - 905; DOI: 10.1021/jm00279a006 |
|
Relative carcinogenicity of some diethylbenz[a]anthracenes J. Pataki and R. Balick pp 905 - 909; DOI: 10.1021/jm00279a007 |
|
14.alpha.,17.alpha.-alkylidenedioxyprogesterone derivatives Dirk Van der Sijde, Herman J. Kooreman, Kapil D. Jaitly, and Arthur F. Marx pp 909 - 914; DOI: 10.1021/jm00279a008 |
|
5-Hydroxy-3-piperidylidenemethane derivatives as spasmolytics Mitsutaka Kawazu, Takeshi Kanno, Seiichi Saito, and Hajime Tamaki pp 914 - 918; DOI: 10.1021/jm00279a009 |
|
Antimalarials. 3. 2,6-Bis(aryl)-4-pyridinemethanols with trifluoromethyl substituents A. Markovac, M. P. LaMontagne, P. Blumbergs, A. B. Ash, and C. L. Stevens pp 918 - 922; DOI: 10.1021/jm00279a010 |
|
Heterocyclic compounds. 10. Synthesis of some imidazo[1,2-a]benzimidazoles with potent analgetic activities Haruo Ogura, Hiroaki Takayanagi, Yukio Yamazaki, Shoichi Yonezawa, Hiromu Takagi, Shinsaku Kobayashi, Toshiharu Kamioka, and Katuo Kamoshita pp 923 - 926; DOI: 10.1021/jm00279a011 |
|
Synthesis and antiprotozoal activity of methylnitro derivatives of 2,2'-biimidazole Piero Melloni, Emanuele Dradi, Willy Logemann, Ivo De Carneri, and Franca Trane pp 926 - 930; DOI: 10.1021/jm00279a012 |
|
Analgetics based on the pyrrolidine ring. 6 Ian M. Lockhart, Nigel E. Webb, Michael Wright, Claude V. Winder, and Pearl Varner pp 930 - 934; DOI: 10.1021/jm00279a013 |
|
5-Substituted-1-indancarboxylic acids as potential antiinflammatory agents George R. Allen, Ruddy Littell, Francis J. McEvoy, and Adolph E. Sloboda pp 934 - 937; DOI: 10.1021/jm00279a014 |
|
Irreversible enzyme inhibitors. 194. Hydrophobic bonding to some dehydrogenases by substituted 5-phenylethyl-4-hydroxyquinoline-3-carboxylic acids B. R. Baker and Ray R. Bramhall pp 937 - 940; DOI: 10.1021/jm00279a015 |
|
Irreversible enzyme inhibitors. 195. Inhibitors of thymidine kinase from Walker 256 carcinoma derived from thymidine 5'-acetate B. R. Baker and John P. Neenan pp 940 - 944; DOI: 10.1021/jm00279a016 |
|
Irreversible enzyme inhibitors. 196. Active-site-directed irreversible inhibitors of dihydrofolate reductase derived from 1-(4-benzyloxy-3-chlorophenyl)-4,6-diamino-1,2-dihydro-2,2-dimethyl-s-triazine and bearing a terminal phenyl sulfonate group B. R. Baker and Wallace T. Ashton pp 945 - 947; DOI: 10.1021/jm00279a017 |
|
Cycloaddition of acetylenes to 7-acylamino-3-azidomethyl-3-cephem-4-carboxylic acids David Willner, Alex M. Jelenevsky, and Lee C. Cheney pp 948 - 951; DOI: 10.1021/jm00279a018 |
|
Schistosomicidal 5-nitro-4-thiazolines Peter J. Islip, Michael D. Closier, Martin C. Neville, Leslie M. Werbel, and David B. Capps pp 951 - 954; DOI: 10.1021/jm00279a019 |
|
1-Alkyl-3-(3-alkyl-5-nitro-4-thiazolin-2-ylidene)ureas and related compounds as schistosomicides Leslie M. Werbel, Margaret B. Degnan, Gail F. Harger, David B. Capps, Peter J. Islip, and Michael D. Closier pp 955 - 963; DOI: 10.1021/jm00279a020 |
|
Metabolic fate of chlorpropamide in man and in the rat Richard C. Thomas and Ray W. Judy pp 964 - 968; DOI: 10.1021/jm00279a021 |
|
Effect of the sulfur-covering group on the antiradiation activity of substituted 2-aminoethanethiols Roger D. Westland, Mary L. Mouk, Joyce L. Holmes, Richard A. Cooley, Jean S. Hong, and Marie M. Grenan pp 968 - 975; DOI: 10.1021/jm00279a022 |
|
Potential antiradiation agents. p-Anisylbutyl derivatives of S-2-aminoethyl hydrogen thiosulfate, 2-aminoethanethiol, the corresponding disulfide, and thiazolidine Roger D. Westland and Joyce L. Holmes pp 976 - 978; DOI: 10.1021/jm00279a023 |
|
L-Asparaginol and derivatives. Synthesis and screening data A. Giner-Sorolla, W. Kreis, C. Gryte, M. L. Cox, and J. H. Burchenal pp 978 - 980; DOI: 10.1021/jm00279a024 |
|
Synthesis and alkylation of tetrahydrofuro[3,4-c]pyrazolols William J. Fanshawe, Victor J. Bauer, and S. R. Safir pp 980 - 982; DOI: 10.1021/jm00279a025 |
|
Imidazo[1,2-a]pyridine anthelmintic and antifungal agents Michael H. Fisher and Aino Lusi pp 982 - 985; DOI: 10.1021/jm00279a026 |
|
Quinazolines and 1,4-benzodiazepines. 55. Synthesis and two metabolites of demoxepam isolated from the dog E. E. Garcia, L. E. Benjamin, R. Ian Fryer, and L. H. Sternbach pp 986 - 987; DOI: 10.1021/jm00279a027 |
|
Antifungal activity of 7- and 5,7-substituted 8-quinolinols Herman Gershon, Maynard W. McNeil, Raulo Parmegiani, and Patricia K. Godfrey pp 987 - 989; DOI: 10.1021/jm00279a028 |
|
Antimalarial potency of 2-benzoyl-4-quinolinemethanols Andrew J. Saggiomo, Shinzo Kano, Toyohiko Kikuchi, Kazumi Okubo, and Masafu Shinbo pp 989 - 994; DOI: 10.1021/jm00279a029 |
|
Absolute configuration of 3-quinuclidinyl benzilate and the behavioral effect in the dog of the optical isomers Anita Meyerhoffer pp 994 - 995; DOI: 10.1021/jm00279a030 |
|
Terpene compounds as drugs. 11. Anabolic 19-nortestosterone terpenoates Gianfranco Pala, Silvano Casadio, Antonio Mantegani, Graziano Bonardi, and Germano Coppi pp 995 - 998; DOI: 10.1021/jm00279a031 |
|
Terpene compounds as drugs. 14. Terpenyl carbamates as central nervous system depressants Giovanna Minoli, Ernesta Marazzi-Uberti, and Silvano Casadio pp 998 - 998; DOI: 10.1021/jm00279a032 |
|
Benzimidazolyl-1,2,4-(H)-triazoles as central nervous system depressants Surendra S. Parmar, A. K. Gupta, H. H. Singh, and T. K. Gupta pp 999 - 1000; DOI: 10.1021/jm00279a033 |
|
Substituted indolebenzylhydrazines as anticonvulsants V. K. Agarwal, T. K. Gupta, and Surendra S. Parmar pp 1000 - 1001; DOI: 10.1021/jm00279a034 |
|
Book Reviews pp 1001 - 1002; DOI: 10.1021/jm00279a600 |
|
gem-Dialkyl effect in medicinal agents Melvin S. Newman, Walter J. J. Broger, Jules B. LaPidus, and Arthur Tye pp 1003 - 1006; DOI: 10.1021/jm00280a001 |
|
Utilization of operational schemes for analog synthesis in drug design John G. Topliss pp 1006 - 1011; DOI: 10.1021/jm00280a002 |
|
Relation of structures and microbiological activities of the 16-membered macrolides Satoshi Omura, Max Tishler, Akira Nakagawa, Yukino Hironaka, and Toju Hata pp 1011 - 1015; DOI: 10.1021/jm00280a003 |
|
Angiotensin II antagonism. Structure-activity relations of 8-substituted angiotensin II analogs D. C. Fessler, F. Sipos, G. S. Denning, D. T. Pals, and F. D. Masucci pp 1015 - 1016; DOI: 10.1021/jm00280a004 |
|
Effect of an amide group in place of the disulfide bridge in deaminooxytocin Satoe Hase, S. Sakakibara, M. Wahrenberg, and Roderich Walter pp 1017 - 1019; DOI: 10.1021/jm00280a005 |
|
Cytotoxic nucleotide analogs as potential anticancer agents. 5-Bromodeoxyuridine 5'-methylphosphonate Paul W. Wigler and Carmen B. Lozzio pp 1020 - 1024; DOI: 10.1021/jm00280a006 |
|
Amidines. 3. Thioureas possessing antihypertensive activity Bernard Loev, Paul E. Bender, Helene Bowman, Anna Helt, Richard McLean, and Timothy Jen pp 1024 - 1027; DOI: 10.1021/jm00280a007 |
|
1-Substituted-3-aminoalkoxy-4,5-cycloalkylpyrazoles with central nervous system depressant activity Beverly S. Barbaz, Harvey I. Chernov, Neville Finch, Heinz W. Gschwend, and Ali Hamdan pp 1027 - 1029; DOI: 10.1021/jm00280a008 |
|
Synthesis and antiinflammatoy activities of .alpha.-methylfluorene-2-acetic acid and related compounds Eric T. Stiller, Patrick A. Diassi, Daniel Gerschutz, Diane Meikle, James Moetz, Pacifico A. Principe, and Seymour D. Levine pp 1029 - 1032; DOI: 10.1021/jm00280a009 |
|
Xanthone-2-carboxylic acids, a new series of antiallergic substances J. R. Pfister, R. W. Ferraresi, I. T. Harrison, W. H. Rooks, A. P. Roszkowski, A. Van Horn, and J. H. Fried pp 1032 - 1035; DOI: 10.1021/jm00280a010 |
|
Antiparasitic nitroimidazoles. 1. 2-Styryl-5-nitroimidazoles William J. Ross, William B. Jamieson, and Max C. McCowen pp 1035 - 1040; DOI: 10.1021/jm00280a011 |
|
Metabolism of 2-(4-chlorophenyl)thiazol-4-ylacetic acid (fenclozic acid) and related compounds by microorganisms Ralph Howe, Ronald H. Moore, Balbir S. Rao, and Alan H. Wood pp 1040 - 1045; DOI: 10.1021/jm00280a012 |
|
Aromatic hydroxylation of lidocaine and mepivacaine in rats and humans J. Thomas and P. Meffin pp 1046 - 1049; DOI: 10.1021/jm00280a013 |
|
Structure-activity relations. 5. Hydrophobic bonding of sulfonamide drugs with serum albumin Toshio Fujita pp 1049 - 1056; DOI: 10.1021/jm00280a014 |
|
Cycloprop[16.alpha.,17.alpha.,]androstanes Kenneth E. Fahrenholtz, Kenneth P. Meyers, and R. W. Kierstead pp 1056 - 1060; DOI: 10.1021/jm00280a015 |
|
Preparation of a number of 5-butylpyrimidine nucleosides E. H. Hamamura, K. Sato, and J. G. Moffatt pp 1061 - 1065; DOI: 10.1021/jm00280a016 |
|
Chance correlations in structure-activity studies using multiple regression analysis John G. Topliss and Robert J. Costello pp 1066 - 1068; DOI: 10.1021/jm00280a017 |
|
Structure-activity correlation for substrates of phenylethanolamine N-methyltransferase (PNMT) Ray W. Fuller and Max M. Marsh pp 1068 - 1069; DOI: 10.1021/jm00280a018 |
|
Are calculated electron populations suitable parameters for multiple regression analyses of biological activity P. R. Andrews pp 1069 - 1072; DOI: 10.1021/jm00280a019 |
|
Novel synthesis of L-(-)-.alpha.-methyl-3,4-dimethoxyphenylalanine Kurt Freter, Manfred Goetz, and Karl Grozinger pp 1072 - 1073; DOI: 10.1021/jm00280a020 |
|
Synthesis of insect-repellent amino analogs of 2-ethyl-1,3-hexanediol (Rutgers 612) Ronald P. Quintana, Paul T. Mui, Andrew Lasslo, Margaret A. Boulware, Carl Schreck, and Harry K. Gouck pp 1073 - 1074; DOI: 10.1021/jm00280a021 |
|
Synthesis of the phosphonic acid isostere of glycerol 3-phosphate Joel Kabak, Louis Defilippe, Robert Engel, and Burton Tropp pp 1074 - 1075; DOI: 10.1021/jm00280a022 |
|
Synthesis and antiviral activity of 4'-hydroxy-5,6,7,8-tetramethoxyflavone Weldon S. Burnham, Robert W. Sidwell, Richard L. Tolman, and Mason G. Stout pp 1075 - 1076; DOI: 10.1021/jm00280a023 |
|
Mechanism of the reaction of a 1,4-benzodiazepine N-oxide with acetic anhydride Neal Castagnoli and Wolfgang Sadee pp 1076 - 1078; DOI: 10.1021/jm00280a024 |
|
2-Benzylaziridines. Cyclic analogs of amphetamines Keith Brewster and Roger M. Pinder pp 1078 - 1079; DOI: 10.1021/jm00280a025 |
|
Central nervous system depressants. 10. 1-Carbamoylbenzodiazepines Robert Bruce Moffett and Allan D. Rudzik pp 1079 - 1081; DOI: 10.1021/jm00280a026 |
|
Derivatives of indole-1-acetic acid as antiinflammatory agents Karl J. Doebel and Jan W. F. Wasley pp 1081 - 1082; DOI: 10.1021/jm00280a027 |
|
Hypotensive thiadiazoles A. M. Grant, S. V. Krees, A. B. Mauger, W. J. Rzeszotarski, and F. W. Wolff pp 1082 - 1084; DOI: 10.1021/jm00280a028 |
|
Carbanilic acid esters of cyclic amino alcohols. 5. Local anesthetic potency of the enantiomers of two N-butyl-3-piperidyl carbanilates Hans Sievertsson, Richard Dahlbom, Rune Sandberg, and Bengt Akerman pp 1085 - 1086; DOI: 10.1021/jm00280a029 |
|
Nitroheterocyclic antimicrobial agents. 1-Methyl-2-nitro-5-imidazolyl derivatives Goro Asato and Gerald Berkelhammer pp 1086 - 1088; DOI: 10.1021/jm00280a030 |
|
Potential antitumor agents. 2. .alpha.- and .beta.-2'-Deoxy-6-selenoguanosine and related compounds Shih-Hsi Chu and Darrell D. Davidson pp 1088 - 1089; DOI: 10.1021/jm00280a031 |
|
Terpene compounds as drugs. 13. o-Terpenylaminomethylphenols and their N-methyl derivatives Arturo Donetti, Silvano Casadio, Cecilia Molino, Graziano Bonardi, and Amedeo Omodei-Sale pp 1089 - 1091; DOI: 10.1021/jm00280a032 |
|
Derivatives of 3,5-dihydro-4H-benzo[2,3]diazepin-4-one K. Nagarajan, J. David, and R. K. Shah pp 1091 - 1092; DOI: 10.1021/jm00280a033 |
|
Synthesis of 9-(3-deoxy-3-fluoro-.beta.-D-arabinofuranosyl)adenine Kenji Miyai, Roland K. Robins, and Richard L. Tolman pp 1092 - 1093; DOI: 10.1021/jm00280a034 |
|
Book reviews pp 1093 - 1094; DOI: 10.1021/jm00280a600 |
|
Oral gold. Antiarthritic properties of alkylphosphinegold coordination complexes Blaine M. Sutton, Elizabeth McGusty, Donald T. Walz, and Michael J. DiMartino pp 1095 - 1098; DOI: 10.1021/jm00281a001 |
|
New substrates for a pancreatic exocrine function test Peter L. DeBenneville, William J. Godfrey, Homer J. Sims, and Anthony R. Imondi pp 1098 - 1100; DOI: 10.1021/jm00281a002 |
|
Conformational and structural relations among antipeptic ulcer compounds Thomas M. Bustard and Yvonne C. Martin pp 1101 - 1105; DOI: 10.1021/jm00281a003 |
|
Semisynthetic .beta.-lactam antibiotics. 1. Acylation of 6-aminopenicillanic acid with activated derivatives of .alpha.-sulfophenylacetic acid Shiro Morimoto, Hiroaki Nomura, Toshihiro Ishiguro, Takeshi Fugono, and Kihachiro Maeda pp 1105 - 1108; DOI: 10.1021/jm00281a004 |
|
Semisynthetic .beta.-lactam antibiotics. 2. Synthesis and properties of D- and L-.alpha.-sulfobenzylpenicillins Shiro Morimoto, Hiroaki Nomura, Takeshi Fugono, Toshiyuki Azuma, Isao Minami, Masatake Hori, and Toru Masuda pp 1108 - 1111; DOI: 10.1021/jm00281a005 |
|
1-Substitutedvinyl-1-phthalanpropylamines as potential antidepressant agents Francis J. McEvoy, Robert F. R. Church, E. N. Greenblatt, and George R. Allen pp 1111 - 1116; DOI: 10.1021/jm00281a006 |
|
p-Substituted N-acetyl-L-(S)- and D(R)-.alpha.-amino-N-phenylsuccinimides and -glutarimides. Substituent effects on stereoselective anticonvulsant activity Donald T. Witiak, Shiv K. Seth, Eugene R. Baizman, Stuart L. Weibel, and Harold H. Wolf pp 1117 - 1123; DOI: 10.1021/jm00281a007 |
|
Cycloalkane spiroheterocyclic compounds. 9. 8-(1,2,3,4-Tetrahydro-2-naphthyl)-2-oxo-1-oxa-3,8-diazaspiro[4,5]decanes and related compounds Jacques Maillard, Michel Langlois, Pierre Delaunay, Vo-Van-Tri, Jacques Chenu, Robert Morin, Marguerite Benharkate, Chantal Manuel, and Francoise Motosso pp 1123 - 1128; DOI: 10.1021/jm00281a008 |
|
Hypocholesterolemic agents. 9. C-20 Epimeric 22,25-diazacholesterols F. Kohen, V. V. Ranade, and R. E. Counsell pp 1129 - 1131; DOI: 10.1021/jm00281a009 |
|
3(2H)-Isoquinolones. 1. 3-Oxygenated analogs of papaverine as peripheral vasodilators William E. Kreighbaum, William F. Kavanaugh, William T. Comer, and David Deitchman pp 1131 - 1135; DOI: 10.1021/jm00281a010 |
|
Antimetabolites of coenzyme Q. 17. Improved synthesis of 5-hydroxy-1,4-benzoquinone analogs and their indices Conny Bogentoft, Alexander Von Klaudy, and Karl Folkers pp 1135 - 1138; DOI: 10.1021/jm00281a011 |
|
Folate antagonists. 9. 2,4-Diamino-6-[(aralkyl)alkylamino]quniazolines, a potent class of antimetabolites with prodigious antimalarial effects Edward F. Elslager, O. D. Bird, Jane Clarke, S. C. Perricone, Donald F. Worth, and John Davoll pp 1138 - 1146; DOI: 10.1021/jm00281a012 |
|
Metabolism of diphenidol. Urinary products in humans and dogs Carl Kaiser, James E. Swagzdis, Thomas L. Flanagan, Bruce M. Lester, Garth L. Burghard, Harry Green, and Charles L. Zirkle pp 1146 - 1150; DOI: 10.1021/jm00281a013 |
|
Design, synthesis, and broad spectrum antiviral activity of 1-.beta.-D-ribofuranosyl-1,2,4-triazole-3-carboxamide and related nucleosides J. T. Witkowski, Roland K. Robins, Robert W. Sidwell, and Lionel N. Simon pp 1150 - 1154; DOI: 10.1021/jm00281a014 |
|
Potential antitumor agents. 6. Possible irreversible inhibitors of ribonucleoside diphosphate reductase Krishna C. Agrawal, Barbara A. Booth, E. Colleen Moore, and Alan C. Sartorelli pp 1154 - 1158; DOI: 10.1021/jm00281a015 |
|
Antitumor and antileukemic effects of some steroids and other biologically interesting compounds containing an alkylating agent F. I. Carroll, Abraham Philip, J. T. Blackwell, D. Jane Taylor, and Monroe E. Wall pp 1158 - 1161; DOI: 10.1021/jm00281a016 |
|
Potential antifertility agents. 3. Substituted dibenzothiophenecarboxylic acids and derivatives R. R. Crenshaw, G. M. Luke, T. A. Jenks, G. Bialy, and M. E. Bierwagen pp 1162 - 1165; DOI: 10.1021/jm00281a017 |
|
Antiandrogens. 2',3'.alpha.-Tetrahydrofuran-2'-spiro-17-(1,2.alpha.-methylene-4-androsten-3-ones) G. H. Rasmusson, A. Chen, G. F. Reynolds, D. J. Patanelli, A. A. Patchett, and G. E. Arth pp 1165 - 1168; DOI: 10.1021/jm00281a018 |
|
Azaindole anthelmintic agents Michael H. Fisher, George Schwartzkopf, and Dale R. Hoff pp 1168 - 1171; DOI: 10.1021/jm00281a019 |
|
Novel cephalosporins. Modification of the carbon-4 carboxyl group Timothy Jen, Barbara Dienel, James Frazee, and Jerry Weisbach pp 1172 - 1174; DOI: 10.1021/jm00281a020 |
|
Iodophenyl derivatives of .alpha.-methyl alanine and isovaline as potential oral cholecystographic agents Gad Shtacher and Shlomo Dayagi pp 1174 - 1177; DOI: 10.1021/jm00281a021 |
|
Preparation and antitumor properties of analogs of acronycine Kenneth J. Liska pp 1177 - 1179; DOI: 10.1021/jm00281a022 |
|
Potential antifertility agents. 2. Tetrazole derivatives of nonsteroidal estrogens R. R. Crenshaw, G. M. Luke, and G. Bialy pp 1179 - 1180; DOI: 10.1021/jm00281a023 |
|
Adamantyl analogs of 2'-(3-dimethylaminopropylthio)cinnamanilide V. L. Narayanan pp 1180 - 1182; DOI: 10.1021/jm00281a024 |
|
Resolution of terbutaline, a new .beta.-sympathomimetic amine K. Wetterlin pp 1182 - 1183; DOI: 10.1021/jm00281a025 |
|
Synthesis and pharmacological actions of 2-[(2-chloroethyl)methylamino]ethyl acetate and some of its derivatives on the isolated guinea pig ileum Clarence Harold Jackson and Maurice Hirst pp 1183 - 1184; DOI: 10.1021/jm00281a026 |
|
Synthesis and biologic activity of p-hydroxylaminopropiophenone Frederick G. DeFeo, Thomas J. Fitzgerald, and John Doull pp 1185 - 1187; DOI: 10.1021/jm00281a027 |
|
Absolute configuration of (+)- and (-)-trans-2-phenylcyclopropylamine hydrochloride Thomas N. Riley and C. G. Brier pp 1187 - 1188; DOI: 10.1021/jm00281a028 |
|
Antimalarial activity of clopidol, 3,5-dichloro-2,6-dimethyl-4-pyridinol, and its esters, carbonates, and sulfonates Lowell D. Markley, John C. Van Heertum, and Harold E. Doorenbos pp 1188 - 1189; DOI: 10.1021/jm00281a029 |
|
N-Alkyl derivatives of purine-6(1H)-thione John A. Montgomery, H. Jeanette Thomas, and Kathleen Hewson pp 1189 - 1192; DOI: 10.1021/jm00281a030 |
|
Medicinal chemistry of (10) annulenes and related compounds. 2. N-(2-Chloroethyl) derivatives of 11-azatricyclo[4.4.1.01,6]undecane, 11-azatricyclo[4.4.1.01,6]undeca-3,8-diene, and 11-azabicyclo[4.4.1]undeca-1,3,5,7,9-pentaene Gary L. Grunewald and Ann M. Warner pp 1192 - 1194; DOI: 10.1021/jm00281a031 |
|
Hydroxylamine derivatives as potential antimalarial agents. 2. Hydroxamates and amidoximes John B. Hynes and Linda G. Hack pp 1194 - 1196; DOI: 10.1021/jm00281a032 |
|
Thiolesters of orotic acid Dale R. Sargent and Charles G. Skinner pp 1196 - 1196; DOI: 10.1021/jm00281a033 |
|
Potential anticancer agents. IV. Schiff bases from benzaldehyde nitrogen mustards D. R. Shekawat, S. S. Sabnis, and C. V. Deliwala pp 1196 - 1197; DOI: 10.1021/jm00281a034 |
|
Prolintane metabolites. Synthesis of dl-1-(.alpha.-propylphenethyl)pyrrolidin-2-one David C. Remy, William A. Van Saun, and Victor J. Lotti pp 1198 - 1198; DOI: 10.1021/jm00281a035 |
|
Hydroxylamine derivatives as potential antimalarial agents. 3. 1,2,4-Oxadiazoles John B. Hynes and Roy F. Gratz pp 1198 - 1200; DOI: 10.1021/jm00281a036 |
|
Book Reviews pp 1200 - 1202; DOI: 10.1021/jm00281a600 |
|
Fused pyrimidines as potential antimicrobic agents Alfred Richardson and Frederick J. McCarty pp 1203 - 1206; DOI: 10.1021/jm00282a001 |
|
Comparative kinetics of cytosine nucleosides. Influence of a 6-methyl substituent on degradation rates and pathways in aqueous buffers Robert E. Notari, Donald T. Witiak, Joyce L. DeYoung, and Ai Jeng Lin pp 1207 - 1214; DOI: 10.1021/jm00282a002 |
|
Synthesis and antitumor antiviral activities of 1-.beta.-D-arabinofuranosylpyrimidine 3',5'-cyclic phosphates Robert A. Long, Gabor L. Szekeres, Tasneem A. Khwaja, Robert W. Sidwell, Lionel N. Simon, and Roland K. Robins pp 1215 - 1218; DOI: 10.1021/jm00282a003 |
|
Pyrimidine nucleosides. 5. Synthesis of carcinostatic halogenocyclonucleosides Tadashi Kanai, Motonobu Ichino, Akio Hoshi, Fumihiko Kanzawa, and Kazuo Kuretani pp 1218 - 1221; DOI: 10.1021/jm00282a004 |
|
Indigogenic phosphodiesters as potential chromogenic cancer chemotherapeutic agents K. C. Tsou, K. W. Lo, S. L. Ledis, and E. E. Miller pp 1221 - 1225; DOI: 10.1021/jm00282a005 |
|
Novel phosphate anthelmintics. 1. Alkyl 2,2-dichlorovinyl methyl phosphates and related alkoxyalkyl and cycloalkyl analogs of dichlorvos Juan G. Morales, Richard H. Whetstone, Donald W. Stoutamire, and D. Kendall Hass pp 1225 - 1231; DOI: 10.1021/jm00282a006 |
|
Novel phosphate anthelmintics. 2. Aralkyl and aralkenyl analogs of dichlorvos John B. Carr, Peter Kirby, Marvin H. Goodrow, Harry G. Durham, D. Kendall Hass, and Judith J. Boudreau pp 1231 - 1234; DOI: 10.1021/jm00282a007 |
|
Partly reduced biphenyls as central nervous system agents. 1. 4-Arylcyclohex-3-enylamines Daniel Lednicer, D. Edward Emmert, Robert Lahti, and Allan D. Rudzik pp 1235 - 1238; DOI: 10.1021/jm00282a008 |
|
Partly reduced biphenyls as central nervous system agents. 2. Cis- and trans-4-arylcyclohexylamines Daniel Lednicer, D. Edward Emmert, Robert Lahti, and Allan D. Rudzik pp 1239 - 1243; DOI: 10.1021/jm00282a009 |
|
Central nervous system agents. 4. Analogs of 3-amino-2-phenylpropiophenone Robert Bruce Moffett and Jackson B. Hester pp 1243 - 1247; DOI: 10.1021/jm00282a010 |
|
Potential bioreductive alkylating agents. 1. Benzoquinone derivatives Ai Jeng Lin, Lucille A. Cosby, Charles W. Shansky, and Alan C. Sartorelli pp 1247 - 1252; DOI: 10.1021/jm00282a011 |
|
Synthesis and antidepressant activity of 5-phenyl-2-(2-propynylamino)-2-oxazolin-4-one and derivatives Cheuk-Man Lee, Bruce W. Horrom, Raymond J. Michaels, Ronald M. Rasmussen, and Nicholas P. Plotnikoff pp 1252 - 1255; DOI: 10.1021/jm00282a012 |
|
Lincomycin. 14. Improved synthesis and resolution of the antimalarial agent, 1'-demethyl-4'-depropyl-4'(R)- and -(S)-pentylclindamycin hydrochloride (U-24, 729A) Barney J. Magerlein pp 1255 - 1259; DOI: 10.1021/jm00282a013 |
|
Synthesis of some histidine analogs and their effect on the growth of a histidine-requiring mutant of Leuconostoc mesenteroides Gordon E. Trout pp 1259 - 1261; DOI: 10.1021/jm00282a014 |
|
Substrate specificity of pyridoxine dehydrogenase from yeast, and the synthesis and biological activities of 5-vinyl and 5-ethynyl analogs of pyridoxol W. Korytnyk, N. Angelino, B. Lachmann, and P. G. G. Potti pp 1262 - 1265; DOI: 10.1021/jm00282a015 |
|
Absolute configurations of the four warfarin alcohols Kenneth K. Chan, Richard J. Lewis, and William F. Trager pp 1265 - 1270; DOI: 10.1021/jm00282a016 |
|
Naphthylalkyl lactamimides as inhibitors of blood platelet aggregation Edward M. Roberts, J. Martin Grisar, Robert D. Mackenzie, George P. Claxton, and Thomas R. Blohm pp 1270 - 1273; DOI: 10.1021/jm00282a017 |
|
Treloxinate and related hypolipidemic 12H-dibenzo[d,g][1,3]dioxocin-6-carboxylate derivatives J. Martin Grisar, Roger A. Parker, Takashi Kariya, Thomas R. Blohm, Robert W. Fleming, and Vladimir Petrow pp 1273 - 1278; DOI: 10.1021/jm00282a018 |
|
Analgesic 1-oxidized-2,6-methano-3-benzazocines William F. Michne and Noel F. Albertson pp 1278 - 1281; DOI: 10.1021/jm00282a019 |
|
17-Aminoacylamido steroid antidepressants George Flouret, Wayne Cole, and Ursula Biermacher pp 1281 - 1283; DOI: 10.1021/jm00282a020 |
|
Inhibition of cholesterol side-chain cleavage. 2. Synthesis of epimeric azacholesterols Matthias C. Lu, P. Afiatpour, C. B. Sullivan, and R. E. Counsell pp 1284 - 1287; DOI: 10.1021/jm00282a021 |
|
Sterols. 38. Synthesis of 1,2.beta.-methylene-17.alpha.-acetoxy-9.beta.,10.alpha.-pregnanes, a class of potent progestational agents S. J. Halkes, J. Hartog, L. Morsink, and A. M. De Wachter pp 1288 - 1292; DOI: 10.1021/jm00282a022 |
|
Sterols. 39. Synthesis and progestational activities of some 16-methylene-17.alpha.-acetoxy-9.beta.,10.alpha.-pregna-4,6-diene-3,20-dione derivatives J. Hartog, J. I. G. M. Wittelaar, L. Morsink, and A. M. De Wachter pp 1292 - 1297; DOI: 10.1021/jm00282a023 |
|
Antiinflammatory activity of some indan-1-carboxylic acids and related compounds P. F. Juby, W. R. Goodwin, T. W. Hudyma, and R. A. Partyka pp 1297 - 1306; DOI: 10.1021/jm00282a024 |
|
Antiinflammatory activity and structure-activity relationships of some 1,2,3,4-tetrahydro-1-naphthoic acids P. F. Juby, W. R. Goodwin, T. W. Hudyma, and R. A. Partyka pp 1306 - 1310; DOI: 10.1021/jm00282a025 |
|
Folic acid analogs. Modifications in the benzene-ring region. 2. Thiazole analogs Eugene C. Roberts and Y. Fulmer Shealy pp 1310 - 1312; DOI: 10.1021/jm00282a026 |
|
2-Mercaptoacetamidine and derivatives as antiradiation agents Roger D. Westland, Mary M. Merz, Susan M. Alexander, Linda S. Newton, Ludwig Bauer, Terry T. Conway, Jerry M. Barton, Krishan K. Khullar, Prabhakar B. Devdhar, and Marie M. Grenan pp 1313 - 1321; DOI: 10.1021/jm00282a027 |
|
Pyridine isosteres of the .beta.-adrenergic antagonists, 2-(p-nitrophenyl)-1-isopropylamino-2-ethanol and 3-(p-nitrophenoxy)-1-isopropylamino-2-propanol C. Thomas Gneuwuch and Harris L. Friedman pp 1321 - 1324; DOI: 10.1021/jm00282a028 |
|
p-Dimethylaminobenzonitrile. Chemically simple coccidiostat Roger C. Parish, Vassilios J. Theodorides, Donald W. Kunkle, Eleanor M. Dietz, and Elva A. Shultis pp 1324 - 1325; DOI: 10.1021/jm00282a029 |
|
Antiinflammatory activity of p-substituted N-benzenesulfonyl derivatives of amino acids Ronald F. Borne, Richard L. Peden, I. W. Waters, Myra Weiner, and Marjorie Walz pp 1325 - 1326; DOI: 10.1021/jm00282a030 |
|
Quaternary 4- (and 5-) azolylpyridazinium salts. New class of oral hypoglycemic agents Gretchen E. Wiegand, Victor J. Bauer, S. R. Safir, D. A. Blickens, and S. J. Riggi pp 1326 - 1328; DOI: 10.1021/jm00282a031 |
|
Synthesis of some cis and trans 2-(substituted amino)cyclohexyl phenyl ketones J. C. Letton, E. Maher, and J. E. Gearien pp 1328 - 1331; DOI: 10.1021/jm00282a032 |
|
Synthesis and biological activity of 2,4-diamino-6- and 7-(1-adamantyl)pteridines J. P. Jonak, S. F. Zakrzewski, L. H. Mead, and L. D. Allshouse pp 1331 - 1332; DOI: 10.1021/jm00282a033 |
|
Synthesis of some bis(2,4-diaminopyrimidines) and bis(2,4-diaminoquinazolines) as potential antimalarial agents John B. Hynes, Roy F. Gratz, and Wallace T. Ashton pp 1332 - 1333; DOI: 10.1021/jm00282a034 |
|
Synthesis of the S-riboside of 5-mercaptouracil, an "S-homolog" of pseudouridine Gabor L. Szekeres and Thomas J. Bardos pp 1333 - 1334; DOI: 10.1021/jm00282a035 |
|
1-Glycosyl derivatives of 5-aminoimidazole-4-carboxamide John A. Montgomery and H. Jeanette Thomas pp 1334 - 1336; DOI: 10.1021/jm00282a036 |
|
Effects of some substituted phenanthrenes on the central nervous system Adolph P. Roszkowski, Margery E. Schuler, and Peter H. Nelson pp 1336 - 1338; DOI: 10.1021/jm00282a037 |
|
Additions and Corrections - Folic Acid Analogs. II. p-{[(2,6-Diamino-8-purinyl)methyl]amino} benzoyl-L-glutamic Acid and Related Compounds L. T. Weinstock, B. F. Grabowski, and C. C. Cheng pp 1341 - 1341; DOI: 10.1021/jm00282a600 |
|
Additions and Corrections - Antibacterial Nitrofuran Derivatives. 4. 5-Nitro-2-furaldehyde Hydrazonium-acethydrazones D. Nardi, E .Massarani, R. Pozzi, and L. Degen pp 1341 - 1341; DOI: 10.1021/jm00282a601 |
|
Additions and Corrections - Structure and Tumor-Promoting Activity of Anthralin (1,8-Dihydroxy-9-anthrone) and Related Compounds A. Segal, C. Katz, and B. L. Van Duuren pp 1341 - 1341; DOI: 10.1021/jm00282a602 |
|
Additions and Corrections - Steroidal Heterocycles. 14. 1,8a-Epoxy-1,4-4a,5,6,7,8,8a-octahydro-2-hydroxynapthalene-3-carbonitrile and Related Compounds H. C. Neumann pp 1341 - 1341; DOI: 10.1021/jm00282a603 |
|
Additions and Corrections - Organic Disulfides and Related Substances. 33. Sodium 4-(2-Acetamidoethyldithio)butanesulfinate and Related Compounds as Antiradiation Drugs. L. Field, and Y. H. Khim pp 1341 - 1341; DOI: 10.1021/jm00282a604 |
|
Additions and Corrections - Synthesis and Biological Activity of Some 5-Substituted 2,4-Diamino-6-alkyl-pyrimidines. 3. J. P. Jonak, S. Zakrzewski, and L. H. Mead pp 1341 - 1341; DOI: 10.1021/jm00282a605 |
|
Additions and Corrections - Studies on the Syntheses of Heterocyclic Compounds. 459. Synthesis of Rescinnamine-Like Compounds as Antihypertensive Agents. T. Kametani, M. Ihara, T. Suzuki, T. Takehashi, R. Iwaki, H. Takei, N. Miyake, M. Yoshida, Y. Hasegawa, and H. Kitagawa pp 1341 - 1341; DOI: 10.1021/jm00282a606 |
|
Additions and Corrections - Book Review of "Arzneimittel: Entwicklung, Wirkung, Darstellung" A. Burger pp 1341 - 1341; DOI: 10.1021/jm00282a607 |
|
Additions and Corrections - Synthesis and Antiprotozoal Activity of Methylnitro Derivatives of 2,2'-Biimidazole. P. Melloni, E. Dradi, W. Logemann, I. de Carneri, and F. Trane pp 1341 - 1341; DOI: 10.1021/jm00282a608 |
|
Additions and Corrections- Antifungal Activity of 7- and 5,7-Substituted 8-Quinolinols. H. Gershon, M. W. McNeil, E. Parmegiani, and P. K . Godfrey pp 1341 - 1341; DOI: 10.1021/jm00282a609 |
|
Book Reviews pp 1339 - 1340; DOI: 10.1021/jm00282a610 |